SCHEMBL8485349

SCHEMBL8485349

Cc1cccc(-c2cn(C3CCN(Cc4ccccc4)CC3)nn2)c1

nearest known ligand 0.78

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
DRD4 P21917 13/20 0.78
DRD2 P14416 11/20 0.78
DRD3 P35462 10/20 0.78
SIGMAR1 Q99720 2/20 0.58
KCNH2 Q12809 1/20 0.58
NAMPT P43490 1/20 0.54
ACHE P22303 1/20 0.49
BACE1 P56817 1/20 0.49
DPP4 P27487 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8484199 0.99 DRD4 (0.77) DRD4DRD2DRD3SIGMAR1KCNH2
SCHEMBL8482373 0.88 DRD4 (1.00) DRD4DRD2DRD3SIGMAR1KCNH2
SCHEMBL8482386 0.87 DRD4 (0.84) DRD4DRD2DRD3SIGMAR1KCNH2
SCHEMBL8480606 0.87 DRD4 (0.62) DRD4DRD2DRD3SIGMAR1KCNH2
Hydrochloric Acid SCHEMBL8484909 0.86 DRD4 (0.82) DRD4DRD2DRD3SIGMAR1KCNH2
Hydrochloric Acid SCHEMBL8480602 0.82 DRD4 (0.56) DRD4DRD2DRD3ACHEBACE1
SCHEMBL8121641 0.81 DRD4 (0.85) DRD4DRD2DRD3SIGMAR1KCNH2
SCHEMBL8482381 0.81 DRD4 (0.72) DRD4DRD2DRD3SIGMAR1KCNH2
Hydrochloric Acid SCHEMBL8484196 0.80 DRD4 (0.70) DRD4DRD2DRD3SIGMAR1KCNH2
SCHEMBL8484752 0.77 GABRA1 (0.46) DRD4DRD2DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5939436-A Five-membered heteroaromatic compounds as dopamine receptor subtype ligands MERCK SHARP & DOHME LTD. (GB) 1999-08-17 US disclosed