SCHEMBL8487363

SCHEMBL8487363

CCc1ncnc(N[C@H]2CC[C@@H](C(C)(C)O)CC2)c1Cl

nearest known ligand 0.37

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CHRM4 P08173 4/20 0.37
PIK3CA P42336 3/20 0.36
MTOR P42345 3/20 0.36
PIM1 P11309 2/20 0.36
IRAK4 Q9NWZ3 4/20 0.36
KDM4E B2RXH2 1/20 0.35
BTK Q06187 3/20 0.35
CYP3A4 P08684 2/20 0.34
CYP2C9 P11712 1/20 0.34
HPGDS O60760 1/20 0.33
FLT3 P36888 1/20 0.33
PIM2 Q9P1W9 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8766710 1.00 CHRM4 (0.37) CHRM4PIK3CAMTORPIM1IRAK4
SCHEMBL7198151 0.90 IRAK4 (0.37) CHRM4IRAK4KDM4EBTKCYP3A4
SCHEMBL8120612 0.90 IRAK4 (0.37) CHRM4IRAK4KDM4EBTKCYP3A4
SCHEMBL8484462 0.88 IRAK4 (0.34) CHRM4IRAK4KDM4EBTKCYP3A4
SCHEMBL8487365 0.84 BTK (0.42) IRAK4KDM4EBTKFLT3
SCHEMBL8486785 0.84 BTK (0.42) IRAK4KDM4EBTKFLT3
SCHEMBL8483434 0.82 BTK (0.43) CHRM4PIK3CAMTORIRAK4KDM4E
SCHEMBL8483437 0.82 BTK (0.43) CHRM4PIK3CAMTORIRAK4KDM4E
SCHEMBL8490025 0.81 IRAK4 (0.45) CHRM4IRAK4KDM4EBTKCYP3A4
SCHEMBL8488399 0.81 IRAK4 (0.39) CHRM4IRAK4KDM4EBTKCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5889012-A INSECTICIDE, ACARICIDES, FUNGICIDES HOECHST-SCHERING AGREVO GMBH (DE) 1999-03-30 US disclosed
EP-0787128-A1 SUBSTITUTED CYCLOALKYLAMINO AND CYCLOALKOXY HETEROCYCLES, PROCESS FOR PREPARING THE SAME AND THEIR USE AS PESTICIDES Hoechst Schering AgrEvo GmbH (DE) 1997-08-06 EP disclosed
WO-1996011913-A1 SUBSTITUTED CYCLOALKYLAMINO AND CYCLOALKOXY HETEROCYCLES, PROCESS FOR PREPARING THE SAME AND THEIR USE AS PESTICIDES HOECHST SCHERING AGREVO GMBH (DE) 1996-04-25 WO disclosed