SCHEMBL8488195

SCHEMBL8488195

FC(F)(F)C(C1CCCCC1)([C@H]1CC[C@@H](Oc2ncc3ccccc3n2)CC1)C(F)(F)F

nearest known ligand 0.36

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HCRTR2 O43614 2/20 0.35
HCRTR1 O43613 1/20 0.35
MKNK2 Q9HBH9 1/20 0.34
HRH4 Q9H3N8 2/20 0.33
CDK4 P11802 2/20 0.33
CDK2 P24941 2/20 0.33
CDK7 P50613 2/20 0.33
CDK9 P50750 2/20 0.33
PDE9A O76083 1/20 0.33
ACACB O00763 3/20 0.32
CDK1 P06493 1/20 0.32
CCNE1 P24864 1/20 0.32
CDK5 Q00535 1/20 0.32
HTR3A P46098 1/20 0.31
PTGS1 P23219 3/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6613792 0.82 CDK4 (0.40) HCRTR2HCRTR1MKNK2HRH4CDK4
SCHEMBL9057676 0.75 L3MBTL1 (0.43) HRH4
SCHEMBL5663343 0.72 PDE9A (0.47) MKNK2PDE9A
SCHEMBL29586318 0.71 PDE9A (0.40) HCRTR2HCRTR1MKNK2HRH4PDE9A
SCHEMBL5463861 0.70 HRH4 (0.51) HRH4CDK2CDK9HTR3A
SCHEMBL2320140 0.68 MKNK2 (0.47) MKNK2PDE9AACACB
SCHEMBL30211008 0.68 MKNK2 (0.47) MKNK2PDE9AACACB
SCHEMBL2320138 0.68 MKNK2 (0.47) MKNK2PDE9AACACB
SCHEMBL1177568 0.66 SLC6A2 (0.52) PDE9AHTR3A
SCHEMBL1177572 0.66 SLC6A2 (0.52) PDE9AHTR3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5889012-A INSECTICIDE, ACARICIDES, FUNGICIDES HOECHST-SCHERING AGREVO GMBH (DE) 1999-03-30 US disclosed