SCHEMBL8488258

SCHEMBL8488258

CNC(=O)c1cccc2c(Nc3cc(N)cc(COC(C)=O)c3)c3ccccc3nc12

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TOP2A P11388 8/20 0.67
TOP2B Q02880 7/20 0.67
PARP1 P09874 4/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2C9 P11712 1/20 0.41
KDM1A O60341 3/20 0.38
MAPT P10636 2/20 0.38
L3MBTL1 Q9Y468 2/20 0.38
POLB P06746 2/20 0.38
RAD52 P43351 2/20 0.38
KMT2A Q03164 2/20 0.38
KDM4E B2RXH2 1/20 0.38
MITF O75030 1/20 0.38
LMNA P02545 1/20 0.38
RECQL P46063 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
HDAC4 P56524 1/20 0.38
HDAC7 Q8WUI4 1/20 0.38
HDAC6 Q9UBN7 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8486786 0.90 TOP2A (0.55) TOP2ATOP2BPARP1CYP3A4CYP2C9
SCHEMBL8488702 0.89 TOP2A (0.67) TOP2ATOP2BPARP1CYP3A4CYP2C9
SCHEMBL8486796 0.88 TOP2A (0.52) TOP2ATOP2BPARP1MAPTKMT2A
SCHEMBL8490361 0.86 TOP2A (0.80) TOP2ATOP2BKDM1AMAPTL3MBTL1
SCHEMBL8489520 0.80 TOP2A (1.00) TOP2ATOP2BKDM1AMAPTL3MBTL1
SCHEMBL8489781 0.79 TOP2A (0.67) TOP2ATOP2BPARP1CYP3A4CYP2C9
SCHEMBL8487444 0.78 TOP2A (0.54) TOP2ATOP2BPARP1CYP3A4CYP2C9
SCHEMBL8489125 0.77 TOP2A (0.66) TOP2ATOP2BPARP1CYP3A4CYP2C9
SCHEMBL9299946 0.76 TOP2A (0.72) TOP2ATOP2BKDM1AMAPTL3MBTL1
SCHEMBL3981533 0.74 TOP2A (0.80) TOP2ATOP2BKDM1AMAPTL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5939428-A ANTITUMOR AGENTS AND ANTIGROWTH AGENTS FOR CELLS NATIONAL HEALTH RESEARCH INSTITUTES (TW) 1999-08-17 US disclosed