SCHEMBL8488702

SCHEMBL8488702

CNC(=O)c1cccc2c(Nc3cc(N)cc(CO)c3)c3ccccc3nc12

nearest known ligand 0.67

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TOP2A P11388 9/20 0.67
TOP2B Q02880 8/20 0.67
PARP1 P09874 3/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2C9 P11712 1/20 0.43
HDAC4 P56524 1/20 0.40
HDAC7 Q8WUI4 1/20 0.40
HDAC6 Q9UBN7 1/20 0.40
HDAC9 Q9UKV0 1/20 0.40
HDAC5 Q9UQL6 1/20 0.40
MAPT P10636 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
KDM1A O60341 3/20 0.39
PIM1 P11309 1/20 0.39
PIM2 Q9P1W9 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8487444 0.89 TOP2A (0.54) TOP2ATOP2BPARP1CYP3A4CYP2C9
SCHEMBL8488258 0.89 TOP2A (0.67) TOP2ATOP2BPARP1CYP3A4CYP2C9
SCHEMBL8489781 0.88 TOP2A (0.67) TOP2ATOP2BPARP1CYP3A4CYP2C9
SCHEMBL8489125 0.87 TOP2A (0.66) TOP2ATOP2BPARP1CYP3A4CYP2C9
SCHEMBL8489010 0.84 TOP2A (0.78) TOP2ATOP2BPARP1CYP3A4CYP2C9
SCHEMBL8489028 0.84 TOP2A (0.73) TOP2ATOP2BKDM1A
SCHEMBL8484693 0.82 TOP2A (0.73) TOP2ATOP2BKDM1A
SCHEMBL29536689 0.82 TOP2A (1.00) TOP2ATOP2BHDAC4HDAC7HDAC6
SCHEMBL1865418 0.82 TOP2A (1.00) TOP2ATOP2BHDAC4HDAC7HDAC6
SCHEMBL3985902 0.81 TOP2A (0.71) TOP2ATOP2BPARP1KDM1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5939428-A ANTITUMOR AGENTS AND ANTIGROWTH AGENTS FOR CELLS NATIONAL HEALTH RESEARCH INSTITUTES (TW) 1999-08-17 US disclosed