SCHEMBL8488352

SCHEMBL8488352

CSc1nccc(-c2c(-c3cccc(C(F)(F)F)c3)nc(C3CCCCN3C(=O)OCc3ccccc3)n2O)n1

nearest known ligand 0.44

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
BTK Q06187 4/20 0.44
CPT2 P23786 1/20 0.40
CPT1A P50416 1/20 0.40
CPT1B Q92523 1/20 0.40
HCRTR1 O43613 1/20 0.40
HCRTR2 O43614 1/20 0.40
TMEM97 Q5BJF2 5/20 0.38
SIGMAR1 Q99720 5/20 0.38
MAPK14 Q16539 5/20 0.37
MAPK13 O15264 4/20 0.37
MAPK12 P53778 4/20 0.37
MAPK11 Q15759 4/20 0.37
MAPK9 P45984 3/20 0.37
TRPV4 Q9HBA0 1/20 0.36
AADAT Q8N5Z0 1/20 0.36
RAF1 P04049 1/20 0.35
F2R P25116 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8485395 0.93 BTK (0.44) BTKCPT2CPT1ACPT1BHCRTR1
SCHEMBL8488861 0.89 BTK (0.43) BTKCPT2CPT1ACPT1BHCRTR1
SCHEMBL6173126 0.87 MAPK14 (0.41) MAPK14MAPK13MAPK12MAPK11MAPK9
SCHEMBL8605126 0.86 BTK (0.46) BTKCPT2CPT1ACPT1BHCRTR1
SCHEMBL8488208 0.85 HCRTR1 (0.47) BTKCPT2CPT1ACPT1BHCRTR1
SCHEMBL8491343 0.84 BTK (0.45) BTKCPT2CPT1ACPT1BTMEM97
SCHEMBL8487384 0.82 BTK (0.45) BTKCPT2CPT1ACPT1BTMEM97
SCHEMBL6172304 0.82 MAPK14 (0.49) BTKMAPK14MAPK13MAPK12MAPK11
SCHEMBL8604095 0.81 BTK (0.47) BTKCPT2CPT1ACPT1BTMEM97
SCHEMBL8603751 0.81 BTK (0.47) BTKCPT2CPT1ACPT1BTMEM97

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5859041-A Substituted imidazoles having cytokine inhibitory activity MERCK & CO., INC. (US) 1999-01-12 US disclosed