SCHEMBL8498013

SCHEMBL8498013

CN1C(=O)C=C[C@@]2(C)C1CC[C@@H]1[C@H]2CC[C@]2(C)C(CNC(=O)CCCc3c[nH]c4ccccc34)CC[C@@H]12

nearest known ligand 0.51

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
AR P10275 6/20 0.50
SRD5A2 P31213 1/20 0.44
KCNH2 Q12809 4/20 0.44
MAPT P10636 1/20 0.43
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8498007 1.00 AR (0.50) ARSRD5A2KCNH2MAPTMEN1
SCHEMBL8499232 0.92 AR (0.51) ARSRD5A2KCNH2
SCHEMBL8499238 0.92 AR (0.51) ARSRD5A2KCNH2
SCHEMBL8497989 0.86 SRD5A1 (0.49) SRD5A2MAPT
SCHEMBL8496497 0.86 SRD5A1 (0.49) SRD5A2MAPT
SCHEMBL8525401 0.81 AR (0.60) ARSRD5A2KCNH2
SCHEMBL8525403 0.81 AR (0.60) ARSRD5A2KCNH2
SCHEMBL8524562 0.81 AR (0.60) ARSRD5A2KCNH2
SCHEMBL8525501 0.81 AR (0.62) ARSRD5A2KCNH2
SCHEMBL8525503 0.81 AR (0.62) ARSRD5A2KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0649431-B1 17-AMINO SUBSTITUTED 4-AZASTEROID 5-ALPHA-REDUCTASE INHIBITORS MERCK & CO INC (US) 1999-08-11 EP claimed
US-5639741-A STEROIDS TREATING SKIN DISORDERS MERCK & CO., INC. (US) 1997-06-17 US claimed
EP-0649431-A4 17-AMINO SUBSTITUTED 4-AZASTEROID 5-G(A)-REDUCTASE INHIBITORS. 1995-05-03 EP claimed
EP-0649431-A1 17-AMINO SUBSTITUTED 4-AZASTEROID 5$g(a)-REDUCTASE INHIBITORS MERCK & CO. INC. (US) 1995-04-26 EP claimed