SCHEMBL8500565

SCHEMBL8500565

Fc1ccc(-c2cnc(NCCCc3ncc[nH]3)nc2-c2ccncc2)cc1.Fc1ccc(-c2cnc(NCCNc3ccccc3)nc2-c2ccncc2)cc1

nearest known ligand 0.44

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 2/20 0.44
NAMPT P43490 16/20 0.43
ADORA1 P30542 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7215175 0.94 NAMPT (0.44) NAMPT
SCHEMBL8503014 0.88 PTGS2 (0.37) PTGS2NAMPTADORA1
SCHEMBL7216105 0.87 PTGS2 (0.54) PTGS2ADORA1
SCHEMBL7210277 0.83 PTGS2 (0.56) PTGS2ADORA1
SCHEMBL7210164 0.81 PTGS2 (0.49) PTGS2ADORA1
Dimethylamine SCHEMBL7210227 0.80 PTGS2 (0.56) PTGS2ADORA1
SCHEMBL7210483 0.80 PTGS2 (0.55) PTGS2ADORA1
SCHEMBL7215116 0.79 PTGS2 (0.58) PTGS2ADORA1
SCHEMBL7210115 0.78 PTGS2 (0.47) PTGS2ADORA1
SCHEMBL27530526 0.78 PTGS2 (0.46) PTGS2ADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0948497-A2 SUBSTITUTED PYRIMIDINE COMPOUNDS AND THEIR USE Amgen inc. (US) 1999-10-13 EP disclosed
WO-1998024782-A2 SUBSTITUTED PYRIMIDINE COMPOUNDS AND THEIR USE AMGEN INC. (US) 1998-06-11 WO disclosed