SCHEMBL8501110

SCHEMBL8501110

COc1cc(OC)c(CCN2CCc3ccccc3C2)c(OC)c1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.62
TDP1 Q9NUW8 1/20 0.56
POLB P06746 1/20 0.55
MEN1 O00255 1/20 0.54
KMT2A Q03164 1/20 0.54
ABCB1 P08183 6/20 0.53
ABCC1 P33527 1/20 0.52
ALDH1A1 P00352 2/20 0.51
MAPT P10636 2/20 0.51
HTT P42858 1/20 0.51
NPSR1 Q6W5P4 1/20 0.51
TAAR1 Q96RJ0 1/20 0.51
HTR1A P08908 1/20 0.51
DRD2 P14416 1/20 0.51
HTR2A P28223 1/20 0.51
SLC6A4 P31645 1/20 0.51
HTR7 P34969 1/20 0.51
HRH1 P35367 1/20 0.51
DRD3 P35462 1/20 0.51
HTR2B P41595 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8498803 0.87 DHCR7 (0.49) KDM4EABCB1ABCC1DRD2DRD3
SCHEMBL8500338 0.85 POLB (0.60) KDM4ETDP1POLBMEN1KMT2A
SCHEMBL8506538 0.85 DHCR7 (0.55) KDM4EPOLBABCB1ABCC1HTR1A
SCHEMBL8490065 0.85 KDM4E (0.77) KDM4ETDP1POLBMEN1KMT2A
SCHEMBL8506904 0.84 TDP1 (0.59) KDM4ETDP1POLBMEN1KMT2A
SCHEMBL8507999 0.83 POLB (0.54) KDM4ETDP1POLBMEN1KMT2A
SCHEMBL8498783 0.82 KDM4E (0.66) KDM4ETDP1POLBMEN1KMT2A
SCHEMBL8504854 0.81 TDP1 (0.54) KDM4ETDP1POLBMEN1KMT2A
SCHEMBL8501315 0.80 SIGMAR1 (0.68) KDM4ETDP1POLBABCB1ABCC1
SCHEMBL8506973 0.79 ABCB1 (0.71) TDP1ABCB1HTR1ADRD3HTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1999024022-A2 ISOQUINOLINE DERIVATIVES FOR TREATING DISORDERS ASSOCIATED WITH 5HT7 RECEPTORS F. HOFFMANN-LA ROCHE AG (CH) 1999-05-20 WO disclosed