SCHEMBL8501398

SCHEMBL8501398

C=CC(C(=O)O)c1ccc(Oc2c(-c3cccc(O)c3)ccc3cc(O)ccc23)cc1

nearest known ligand 0.51

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 18/20 0.51
ESR2 Q92731 17/20 0.51
AKR1C3 P42330 1/20 0.39
AKR1C2 P52895 1/20 0.39
THRA P10827 1/20 0.36
THRB P10828 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
HSD17B1 P14061 1/20 0.36
CYP2B6 P20813 1/20 0.36
CYP2C19 P33261 1/20 0.36
HSD17B2 P37059 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8497567 0.94 ESR1 (0.43) ESR1ESR2
SCHEMBL8501285 0.91 ESR1 (0.48) ESR1ESR2
SCHEMBL8498119 0.87 ESR1 (0.43) ESR1ESR2CYP3A4CYP2D6CYP2C9
SCHEMBL8497265 0.87 ESR1 (0.52) ESR1ESR2
SCHEMBL8500302 0.85 AKR1C3 (0.45) AKR1C3AKR1C2THRATHRBCYP1A2
SCHEMBL8501030 0.85 AKR1C3 (0.54) ESR1ESR2AKR1C3AKR1C2CYP1A2
SCHEMBL8500328 0.83 AKR1C3 (0.42) ESR1ESR2AKR1C3AKR1C2CYP1A2
SCHEMBL8500430 0.82 PPARG (0.39) ESR1ESR2AKR1C3AKR1C2CYP2C9
SCHEMBL8502302 0.82 ESR1 (0.53) ESR1ESR2AKR1C3AKR1C2
SCHEMBL14615054 0.81 ESR1 (0.65) ESR1ESR2CYP1A2CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5916916-A USEFUL AS SELECTIVE ESTROGEN RECEPTOR MODULATORS. ELI LILLY AND COMPANY (US) 1999-06-29 US claimed
US-5916916-A USEFUL AS SELECTIVE ESTROGEN RECEPTOR MODULATORS. ELI LILLY AND COMPANY (US) 1999-06-29 US disclosed