SCHEMBL8501657

SCHEMBL8501657

COc1cc2c(C3C(=O)Nc4ccccc43)ncnc2cc1OCCc1ncc[nH]1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 1/20 0.37
PDE4B Q07343 1/20 0.37
PDE4C Q08493 1/20 0.37
PDE4D Q08499 1/20 0.37
TNKS O95271 1/20 0.37
PARP1 P09874 1/20 0.37
TNKS2 Q9H2K2 1/20 0.37
EGFR P00533 2/20 0.36
BRD4 O60885 1/20 0.36
ERBB2 P04626 1/20 0.36
ERBB4 Q15303 1/20 0.36
KDR P35968 7/20 0.36
ENPP1 P22413 1/20 0.35
HDAC3 O15379 2/20 0.34
HDAC4 P56524 2/20 0.34
HDAC1 Q13547 2/20 0.34
HDAC7 Q8WUI4 2/20 0.34
HDAC2 Q92769 2/20 0.34
HDAC10 Q969S8 2/20 0.34
HDAC11 Q96DB2 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8501633 0.99 PDE4A (0.37) PDE4APDE4BPDE4CPDE4DTNKS
SCHEMBL6671698 0.89 KDR (0.35) EGFRBRD4ERBB2ERBB4KDR
SCHEMBL6588693 0.87 CHEK1 (0.42) EGFRKDR
SCHEMBL7205793 0.86 KDR (0.48) KDR
SCHEMBL7205653 0.85 PDE4A (0.45) PDE4APDE4BPDE4CPDE4DTNKS
Acetic Acid SCHEMBL4677365 0.84 EGFR (0.36) EGFRKDRENPP1HDAC3HDAC4
SCHEMBL7206414 0.83 KDR (0.46) KDR
Hydrochloric Acid SCHEMBL7211167 0.82 KDR (0.45) KDR
SCHEMBL7209978 0.82 IRAK1 (0.50) EGFRKDRMAPK1ATM
Hydrochloric Acid SCHEMBL8187414 0.82 KDR (0.34) KDRENPP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0912557-A1 OXINDOLE DERIVATIVES ZENECA LIMITED (GB) 1999-05-06 EP disclosed
WO-1997042187-A1 OXINDOLE DERIVATIVES ZENECA LIMITED (GB) 1997-11-13 WO disclosed