SCHEMBL8507705

SCHEMBL8507705

CCCCc1ncc(C=O)n1Cc1ccc(C(=O)OCC)cc1

nearest known ligand 0.64

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
AGTR1 P30556 13/20 0.56
AGTR2 P50052 4/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27406325 0.93 AGTR1 (0.55) AGTR1AGTR2
SCHEMBL27382399 0.92 AGTR1 (0.54) AGTR1AGTR2
SCHEMBL9124156 0.90 AGTR1 (0.49) AGTR1AGTR2
SCHEMBL946900 0.90 AGTR1 (0.67) AGTR1AGTR2
SCHEMBL27532043 0.90 AGTR1 (0.53) AGTR1AGTR2
SCHEMBL27535439 0.88 AGTR1 (0.53) AGTR1AGTR2
SCHEMBL27452523 0.88 AGTR1 (0.52) AGTR1AGTR2
SCHEMBL27405616 0.87 AGTR1 (0.54) AGTR1AGTR2
SCHEMBL951175 0.86 AGTR1 (0.66) AGTR1AGTR2
SCHEMBL7268950 0.86 AGTR1 (0.45) AGTR1AGTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0662961-B1 PROCESS OF SYNTHESIZING USEFUL INTERMEDIATES OF SUBSTITUTED IMIDAZOLE COMPOUNDS SMITHKLINE BEECHAM CORP (US) 1999-11-10 EP claimed
US-5565577-A Process for preparing 1-alkyaryl-2-alkyl-5-formylimidazole SMITHKLINE BEECHAM CORPORATION (US) 1996-10-15 US claimed
EP-0662961-A4 PROCESS OF SYNTHESIZING USEFUL INTERMEDIATES OF SUBSTITUTED IMIDAZOLE COMPOUNDS. SMITHKLINE BEECHAM CORP (US) 1996-07-31 EP claimed
EP-0662961-A1 PROCESS OF SYNTHESIZING USEFUL INTERMEDIATES OF SUBSTITUTED IMIDAZOLE COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 1995-07-19 EP claimed
WO-1994006776-A1 PROCESS OF SYNTHESIZING USEFUL INTERMEDIATES OF SUBSTITUTED IMIDAZOLE COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 1994-03-31 WO claimed
US-5389661-A Treats hypertension, heart failure, glaucoma and hyperaldosteronism WARNER-LAMBERT COMPANY (US) 1995-02-14 US disclosed
US-5322950-A Treating hypertension, hyperaldosteronism, glaucoma, heart failure WARNER-LAMBERT COMPANY (US) 1994-06-21 US disclosed
CN-1081438-A Imdazole derivatives and preparation method thereof and the application on therapeutics FOURNIER IND & SANTE (FR) 1994-02-02 CN disclosed