SCHEMBL8508409

SCHEMBL8508409

COc1cc(C(=O)CCCN2CC[C@@H](OC(=O)c3cc(Cl)c(N)c4c3OCC4)[C@@H](OC)C2)cc(OC)c1OC

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR4 Q13639 5/20 0.49
HTR3A P46098 4/20 0.49
ADRA1A P35348 3/20 0.49
ADRA2C P18825 2/20 0.49
KCNH2 Q12809 2/20 0.49
HTR1A P08908 1/20 0.49
ACHE P22303 1/20 0.49
PTGS1 P23219 1/20 0.49
HTR2C P28335 3/20 0.41
HTR3E A5X5Y0 2/20 0.41
HTR3B O95264 2/20 0.41
HTR3D Q70Z44 2/20 0.41
HTR3C Q8WXA8 2/20 0.41
ADRA2A P08913 2/20 0.41
HTR2A P28223 2/20 0.41
CHRM2 P08172 1/20 0.41
CHRM1 P11229 1/20 0.41
DRD2 P14416 1/20 0.41
ADRA2B P18089 1/20 0.41
CHRM3 P20309 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8508414 1.00 HTR4 (0.49) HTR4HTR3AADRA1AADRA2CKCNH2
SCHEMBL8508412 1.00 HTR4 (0.49) HTR4HTR3AADRA1AADRA2CKCNH2
SCHEMBL8509382 0.89 HTR4 (0.54) HTR4HTR3AADRA1AADRA2CKCNH2
Oxalic Acid SCHEMBL8510621 0.87 HTR4 (0.52) HTR4HTR3AADRA1AADRA2CKCNH2
SCHEMBL8508804 0.85 HTR4 (0.49) HTR4HTR3AADRA1AADRA2CKCNH2
SCHEMBL13036098 0.84 HTR4 (0.52) HTR4HTR3AADRA1AADRA2CKCNH2
SCHEMBL8497984 0.84 HTR4 (0.53) HTR4HTR3AADRA1AADRA2CKCNH2
SCHEMBL8497978 0.84 HTR4 (0.53) HTR4HTR3AADRA1AADRA2CKCNH2
SCHEMBL8943232 0.83 HTR4 (0.52) HTR4HTR3AADRA1AADRA2CKCNH2
SCHEMBL8943236 0.83 HTR4 (0.52) HTR4HTR3AADRA1AADRA2CKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0784619-B1 PHENYL-OXO-ALKYL-(4-PIPERIDINYL)BENZOATE DERIVATIVES JANSSEN PHARMACEUTICA NV (BE) 1999-03-24 EP claimed
EP-0784619-B1 PHENYL-OXO-ALKYL-(4-PIPERIDINYL)BENZOATE DERIVATIVES JANSSEN PHARMACEUTICA NV (BE) 1999-03-24 EP disclosed