SCHEMBL8511378

SCHEMBL8511378

CC(C)(C)OC(=O)NC1(c2ccc(-c3cccc(-c4ccc5c(c4)C(C)(C)CCC5(C)C)n3)cc2)CCC1

nearest known ligand 0.54

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
RARB P10826 5/20 0.54
RARA P10276 4/20 0.54
AKT1 P31749 2/20 0.45
AKT2 P31751 1/20 0.45
RARG P13631 5/20 0.43
PDE2A O00408 5/20 0.36
RXRA P19793 3/20 0.36
CNR1 P21554 1/20 0.36
CNR2 P34972 1/20 0.36
KIT P10721 1/20 0.36
ABCB1 P08183 1/20 0.36
ABCC1 P33527 1/20 0.36
SCN9A Q15858 1/20 0.35
RXRB P28702 1/20 0.35
TACR3 P29371 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8515775 0.86 RARA (0.64) RARBRARAAKT1RARGRXRA
SCHEMBL8512225 0.80 RARA (0.56) RARBRARAAKT1RARG
SCHEMBL17040898 0.73 SSTR4 (0.47) AKT1AKT2CNR1CNR2TACR3
SCHEMBL8515374 0.73 RARB (0.60) RARBRARAAKT1AKT2RARG
SCHEMBL17109509 0.72 AKT1 (0.43) AKT1AKT2PDE2ACNR1CNR2
SCHEMBL14161397 0.72 AKT1 (0.42) AKT1AKT2PDE2ACNR1CNR2
Hydrochloric Acid SCHEMBL8612658 0.72 RARA (0.58) RARBRARAAKT1AKT2RARG
Hydrochloric Acid SCHEMBL8514603 0.72 RARA (0.58) RARBRARAAKT1AKT2RARG
SCHEMBL12633283 0.71 AURKA (0.53) RARBRARA
SCHEMBL25156379 0.71 AKT1 (0.51) AKT1AKT2PDE2ACNR1CNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012069852-A1 PHARMACEUTICAL COMPOUNDS AS INHIBITORS OF SPHINGOSINE KINASE ALMAC DISCOVERY LIMITED (GB) 2012-05-31 WO disclosed