SCHEMBL8511634

SCHEMBL8511634

CC(C)(C)OC(=O)N1CCC2(CCN(c3ccnc(Cl)c3)CC2)C1

nearest known ligand 0.53

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 1/20 0.53
SCD5 Q86SK9 1/20 0.48
ACACB O00763 5/20 0.45
HIF1A Q16665 2/20 0.45
EIF2AK4 Q9P2K8 1/20 0.44
HDAC2 Q92769 1/20 0.43
CYP2C9 P11712 3/20 0.43
CYP3A4 P08684 3/20 0.43
CYP2D6 P10635 2/20 0.43
JAK2 O60674 1/20 0.42
JAK1 P23458 1/20 0.42
RET P07949 1/20 0.42
TSHR P16473 2/20 0.42
POLB P06746 1/20 0.42
ALDH1A1 P00352 1/20 0.41
CYP2C19 P33261 1/20 0.41
GPR183 P32249 1/20 0.41
GPR119 Q8TDV5 1/20 0.40
USP30 Q70CQ3 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21434155 0.86 EGLN2 (0.48) CYP11B2SCD5EIF2AK4JAK2JAK1
SCHEMBL485242 0.85 CYP11B2 (0.51) CYP11B2SCD5ACACBHIF1AEIF2AK4
SCHEMBL1432796 0.85 POLB (0.53) TSHRPOLBALDH1A1GPR119
SCHEMBL484102 0.84 HIF1A (0.63) CYP11B2HIF1ACYP2C9CYP3A4CYP2D6
SCHEMBL20468942 0.83 CYP3A4 (0.50) CYP11B2SCD5ACACBHIF1ACYP2C9
SCHEMBL484886 0.82 CYP11B2 (0.55) CYP11B2SCD5HDAC2CYP2C9CYP3A4
SCHEMBL20468955 0.81 CYP3A4 (0.51) CYP11B2SCD5ACACBHIF1ACYP2C9
SCHEMBL20025395 0.81 EIF2AK4 (0.44) SCD5EIF2AK4JAK2JAK1POLB
SCHEMBL8511358 0.80 CYP11B2 (0.46) CYP11B2SCD5ACACBHIF1AHDAC2
SCHEMBL30328547 0.80 CYP11B2 (0.48) CYP11B2SCD5ACACBHIF1AEIF2AK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012069852-A1 PHARMACEUTICAL COMPOUNDS AS INHIBITORS OF SPHINGOSINE KINASE ALMAC DISCOVERY LIMITED (GB) 2012-05-31 WO disclosed