SCHEMBL8513639

SCHEMBL8513639

NC1CCN(c2ccnc(Br)c2)CC1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 2/20 0.47
HRH4 Q9H3N8 6/20 0.45
AKT2 P31751 3/20 0.42
DKK1 O94907 1/20 0.41
VCP P55072 1/20 0.38
HTR3E A5X5Y0 1/20 0.37
MEN1 O00255 1/20 0.37
HTR3B O95264 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP2D6 P10635 1/20 0.37
ALOX15 P16050 1/20 0.37
TSHR P16473 1/20 0.37
NFKB1 P19838 1/20 0.37
HTR3A P46098 1/20 0.37
KMT2A Q03164 1/20 0.37
HTR3D Q70Z44 1/20 0.37
HTR3C Q8WXA8 1/20 0.37
PAK4 O96013 2/20 0.37
PAK1 Q13153 2/20 0.37
KIT P10721 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21590373 0.81 HRH3 (0.53) HRH3HRH4AKT2DKK1VCP
SCHEMBL1634508 0.80 CHKA (0.52) HRH4MEN1ALOX15KMT2A
SCHEMBL30900615 0.80 CHKA (0.52) HRH4MEN1ALOX15KMT2A
SCHEMBL25247515 0.80 HRH4 (0.47) HRH4
SCHEMBL7008838 0.80 HRH4 (0.48) HRH3HRH4AKT2DKK1KIT
SCHEMBL2272239 0.80 HTR3E (0.47) HRH3HRH4AKT2DKK1VCP
SCHEMBL29132185 0.80 HRH4 (0.35) HRH4CDK1CDK2
SCHEMBL16684915 0.80 SMARCA2 (0.47) HRH3HRH4
SCHEMBL31341814 0.79 HRH4 (0.54) HRH4MEN1ALOX15KMT2A
SCHEMBL5314278 0.79 HRH4 (0.54) HRH4MEN1ALOX15KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012069852-A1 PHARMACEUTICAL COMPOUNDS AS INHIBITORS OF SPHINGOSINE KINASE ALMAC DISCOVERY LIMITED (GB) 2012-05-31 WO disclosed