SCHEMBL8514972

SCHEMBL8514972

CCCc1ccc(Cc2ccc(OC(F)(F)F)cc2)cc1F

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 4/20 0.46
TSHR P16473 1/20 0.41
DAO P14920 1/20 0.41
MPO P05164 1/20 0.39
CYP11B1 P15538 1/20 0.39
CYP11B2 P19099 1/20 0.39
ALDH1A1 P00352 1/20 0.38
ALOX5 P09917 1/20 0.38
CNR2 P34972 1/20 0.38
LMNA P02545 1/20 0.38
SLC6A3 Q01959 3/20 0.37
GPR84 Q9NQS5 1/20 0.36
SLC5A1 P13866 1/20 0.36
SLC5A2 P31639 1/20 0.36
TRPV1 Q8NER1 1/20 0.36
PDE2A O00408 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23055180 0.84 PDE2A (0.47) TSHRLMNATRPV1PDE2A
SCHEMBL8990775 0.82 DAO (0.41) SLC6A4TSHRDAOALDH1A1SLC6A3
SCHEMBL8515213 0.81 SLC6A4 (0.47) SLC6A4TSHRDAOCYP11B1CYP11B2
SCHEMBL9061734 0.79 TSHR (0.43) SLC6A4TSHRDAOALDH1A1LMNA
SCHEMBL7851561 0.78 FFAR1 (0.45) LMNA
SCHEMBL1687455 0.77 TSHR (0.53) SLC6A4TSHRDAOALDH1A1LMNA
SCHEMBL7654059 0.77 TAAR1 (0.40) ALDH1A1ALOX5CNR2LMNA
SCHEMBL2092054 0.77 SLC6A4 (0.56) SLC6A4TSHRDAOMPOCYP11B1
SCHEMBL14959716 0.76 ADRB2 (0.44) MPOLMNATRPV1PDE2A
SCHEMBL8990665 0.76 S1PR1 (0.44) TSHRDAOALDH1A1GPR84

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012069856-A1 ANTIMALARIAL COMPOUNDS LIVERPOOL SCHOOL OF TROPICAL MEDICINE (GB) 2012-05-31 WO disclosed