SCHEMBL8515485

SCHEMBL8515485

CC(C)(C)OC(=O)NC1SCC2(c3cc(Br)ccc3OC3CCCCC32)N1O

nearest known ligand 0.34

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 5/20 0.34
AKR1B1 P15121 3/20 0.33
CTSD P07339 1/20 0.33
CACNA1B Q00975 1/20 0.31
AAK1 Q2M2I8 3/20 0.31
KMT2A Q03164 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
USP30 Q70CQ3 2/20 0.31
RORC P51449 2/20 0.30
SYK P43405 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8515572 0.71 BACE1 (0.40) BACE1AKR1B1CTSDAAK1RORC
SCHEMBL9932816 0.71 BACE1 (0.40) BACE1AKR1B1CTSDAAK1
SCHEMBL876606 0.67 AKR1B1 (0.43) BACE1AKR1B1CTSD
SCHEMBL877188 0.64 AKR1B1 (0.46) BACE1AKR1B1CTSD
SCHEMBL9932213 0.63 BACE1 (0.38) BACE1CTSDAAK1RORC
SCHEMBL877606 0.63 BACE1 (0.45) BACE1AKR1B1CTSD
SCHEMBL8513209 0.62 BACE1 (0.35) BACE1AKR1B1CTSDAAK1
SCHEMBL8613061 0.60 AKR1B1 (0.42) BACE1AKR1B1CTSD
SCHEMBL8613068 0.60 AKR1B1 (0.42) BACE1AKR1B1CTSD
SCHEMBL4146006 0.60 AAK1 (0.41) BACE1CTSDAAK1USP30

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012071458-A1 HETEROCYCLIC INHIBITORS OF BETA - SECRETASE FOR THE TREATMENT OF NEURODEGENERATIVE DISEASES ARRAY BIOPHARMA INC. (US) 2012-05-31 WO disclosed