SCHEMBL8515489

SCHEMBL8515489

COc1ccc(-c2cc(Nc3cccc(NS(C)(=O)=O)c3)ncn2)cc1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCNT1 O60563 5/20 0.68
CDK9 P50750 5/20 0.68
MAP4K4 O95819 1/20 0.68
CDK1 P06493 1/20 0.68
CDK4 P11802 1/20 0.68
CCNB1 P14635 1/20 0.68
CCND1 P24385 1/20 0.68
ABL2 P42684 1/20 0.68
GSK3A P49840 1/20 0.68
CDK7 P50613 1/20 0.68
CCNH P51946 1/20 0.68
MNAT1 P51948 1/20 0.68
CYP1A2 P05177 4/20 0.66
CYP3A4 P08684 4/20 0.66
CYP2C19 P33261 4/20 0.66
CYP2C9 P11712 3/20 0.66
CYP2D6 P10635 3/20 0.66
USP2 O75604 2/20 0.66
CLK4 Q9HAZ1 2/20 0.66
TSHR P16473 1/20 0.66

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8516577 0.87 CYP1A2 (0.86) CCNT1CDK9MAP4K4CDK1CDK4
SCHEMBL8516573 0.86 CYP1A2 (0.69) CCNT1CDK9MAP4K4CDK1CDK4
SCHEMBL4102091 0.84 BACE1 (0.77) CCNT1CDK9MAP4K4CDK1CDK4
SCHEMBL12984174 0.84 CCNT1 (0.60) CCNT1CDK9MAP4K4CDK1CDK4
SCHEMBL4104594 0.83 CCNT1 (0.69) CCNT1CDK9ABL1BCRMEN1
SCHEMBL17022942 0.82 CYP1A2 (0.69) CCNT1CDK9MAP4K4CDK1CDK4
SCHEMBL8514144 0.81 CYP1A2 (0.69) CCNT1CDK9MAP4K4CDK1CDK4
SCHEMBL4107964 0.81 CDK5 (0.62) CCNT1CDK9ABL1BCRMEN1
SCHEMBL4437118 0.81 CCNT1 (0.70) CCNT1CDK9MAP4K4CDK1CDK4
SCHEMBL4109231 0.81 CCNT1 (0.77) CCNT1CDK9MAP4K4CDK1CDK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2137166-B1 4, 6-DISUBSTITUTED AMINOPYRIMIDINE DERIVATIVES AS INHIBITORS OF PROTEIN KINASES INGENIUM PHARMACEUTICALS GMBH (DE) 2012-05-30 EP claimed