SCHEMBL8515827

SCHEMBL8515827

COc1cc(OC)c2c(=O)cc(-c3ccccc3Cl)oc2c1C1CCNC1CCO

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A1 P04798 3/20 0.49
CYP1A2 P05177 3/20 0.49
CYP1B1 Q16678 3/20 0.49
CDK4 P11802 12/20 0.48
CDK1 P06493 11/20 0.48
CCND1 P24385 10/20 0.48
CDK9 P50750 9/20 0.48
CDK2 P24941 8/20 0.48
CCNB1 P14635 8/20 0.48
CCNT1 O60563 7/20 0.48
CCNB2 O95067 6/20 0.48
CCNB3 Q8WWL7 6/20 0.48
CCNA2 P20248 5/20 0.48
CCNE1 P24864 4/20 0.48
GSK3A P49840 4/20 0.48
CCND3 P30281 3/20 0.48
CDK6 Q00534 3/20 0.48
CDK7 P50613 3/20 0.48
CCNH P51946 2/20 0.48
MNAT1 P51948 2/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16722415 0.84 CDK4 (0.64) CDK4CDK1CCND1CDK9CDK2
SCHEMBL291158 0.84 CDK4 (0.64) CDK4CDK1CCND1CDK9CDK2
Hydrochloric Acid SCHEMBL6120022 0.83 CDK4 (0.62) CDK4CDK1CCND1CDK9CDK2
Hydrochloric Acid SCHEMBL17294474 0.83 CDK4 (0.62) CDK4CDK1CCND1CDK9CDK2
SCHEMBL1180448 0.82 CDK4 (0.53) CYP1A1CYP1A2CYP1B1CDK4CDK1
SCHEMBL1180446 0.82 CDK4 (0.53) CYP1A1CYP1A2CYP1B1CDK4CDK1
SCHEMBL14694316 0.82 CYP1A1 (0.42) CYP1A1CYP1A2CYP1B1CDK4CDK1
SCHEMBL291053 0.79 CDK4 (0.75) CYP1A1CYP1A2CYP1B1CDK4CDK1
SCHEMBL291051 0.79 CDK4 (0.75) CYP1A1CYP1A2CYP1B1CDK4CDK1
SCHEMBL6524830 0.79 CDK4 (0.75) CYP1A1CYP1A2CYP1B1CDK4CDK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012069972-A1 A PHARMACEUTICAL COMBINATION FOR THE TREATMENT OF BREAST CANCER PIRAMAL LIFE SCIENCES LIMITED (IN) 2012-05-31 WO disclosed