SCHEMBL8517140

SCHEMBL8517140

C=CCc1ccc2nc(C#CC(C)O)cnc2c1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.36
KDM4E B2RXH2 2/20 0.36
MEN1 O00255 2/20 0.36
GAA P10253 2/20 0.36
MAPT P10636 2/20 0.36
KMT2A Q03164 2/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
LMNA P02545 1/20 0.36
HTT P42858 1/20 0.36
XDH P47989 1/20 0.34
PPARG P37231 2/20 0.33
PPARD Q03181 2/20 0.33
GABRA1 P14867 2/20 0.33
GABRB2 P47870 2/20 0.33
ALDH2 P05091 1/20 0.33
AKR1B1 P15121 1/20 0.33
HPGD P15428 1/20 0.33
CNR1 P21554 1/20 0.33
CNR2 P34972 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8517796 0.81 CYP2D6 (0.43) ALDH1A1MEN1GAAMAPTKMT2A
SCHEMBL8517808 0.78 ALDH1A1 (0.36) ALDH1A1KDM4EMEN1GAAMAPT
SCHEMBL8598799 0.78
SCHEMBL8518290 0.76 EGFR (0.34) PGK1
SCHEMBL8517840 0.74 ACACB (0.41) ALDH1A1KDM4EMEN1GAAMAPT
SCHEMBL8518327 0.73 ACACB (0.40) ALDH1A1KDM4EMEN1GAAMAPT
SCHEMBL8517544 0.71 ALDH1A1 (0.41) ALDH1A1KDM4EMEN1GAAMAPT
SCHEMBL8036653 0.69 ALDH1A1 (0.33) ALDH1A1KDM4EMEN1GAAMAPT
SCHEMBL8036646 0.69 ALDH1A1 (0.33) ALDH1A1KDM4EMEN1GAAMAPT
SCHEMBL8517235 0.69 CYP2D6 (0.38) ALDH1A1KDM4EMEN1MAPTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0628530-B1 ACETYLENE DERIVATIVES, PROCESS FOR PRODUCING THE SAME, LIQUID CRYSTAL COMPOSITION CONTAINING THE SAME AS ACTIVE INGREDIENT, AND LIQUID CRYSTAL ELEMENT MADE THEREFROM SUMITOMO CHEMICAL CO (JP) 1999-03-24 EP disclosed
US-5534188-A Acetylene derivatives, process for producing the same, liquid crystal composition containing the same as an active ingredient, and liquid crystal element using said liquid crystal composition SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1996-07-09 US disclosed
EP-0628530-A1 ACETYLENE DERIVATIVE, PROCESS FOR PRODUCING THE SAME, LIQUID CRYSTAL COMPOSITION CONTAINING THE SAME AS ACTIVE INGREDIENT, AND LIQUID CRYSTAL ELEMENT MADE THEREFROM SUMITOMO CHEMICAL COMPANY LIMITED (JP) 1994-12-14 EP disclosed