SCHEMBL8517516

SCHEMBL8517516

COS(=O)(=O)[O-].C[S+](C)c1ccc(OC(=O)OCc2ccccc2)cc1

nearest known ligand 0.43

Known targets — ChEMBL curated mechanism

ACHECHRM1CHRM3

The experimentally established mechanism targets of None. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE known ✓ P22303 1/20 0.38
KMT2A Q03164 2/20 0.43
MEN1 O00255 1/20 0.43
HTT P42858 1/20 0.43
GFER P55789 1/20 0.43
HSD17B10 Q99714 1/20 0.43
HTR2A P28223 1/20 0.40
ALDH1A1 P00352 3/20 0.40
LMNA P02545 1/20 0.40
MAPT P10636 1/20 0.38
CA1 P00915 2/20 0.38
CA2 P00918 2/20 0.38
TSHR P16473 1/20 0.37
CA12 O43570 1/20 0.36
CA9 Q16790 1/20 0.36
HTR2C P28335 1/20 0.36
MMP13 P45452 2/20 0.36
MMP1 P03956 1/20 0.36
MMP3 P08254 1/20 0.36
MMP7 P09237 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10590429 0.90 HTR2A (0.43) HTTHTR2AALDH1A1MMP1MMP9
SCHEMBL9646440 0.90 KMT2A (0.50) KMT2AMEN1HTTGFERHSD17B10
SCHEMBL30335697 0.85 KMT2A (0.46) KMT2AMEN1HTTGFERHSD17B10
SCHEMBL10590135 0.83 CA1 (0.44) KMT2AMEN1ALDH1A1LMNACA1
SCHEMBL9574220 0.83 CA1 (0.44) KMT2AMEN1ALDH1A1LMNACA1
SCHEMBL6839788 0.82 KMT2A (0.55) KMT2AMEN1HSD17B10ALDH1A1LMNA
SCHEMBL9352481 0.81 ALDH1A1 (0.41) HTTHTR2AALDH1A1MMP1MMP9
SCHEMBL9574203 0.81 ALDH1A1 (0.49) KMT2AMEN1HTTALDH1A1LMNA
SCHEMBL10591248 0.81 ALDH1A1 (0.49) KMT2AMEN1HTTALDH1A1LMNA
SCHEMBL7669154 0.80 KMT2A (0.49) KMT2AMEN1HTTGFERHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0331988-A1 Sulfonium compounds, as well as process for producing active esters and amides used for the production of amides SANSHIN KAGAKU KOGYO CO., LTD. (JP) 1989-09-13 EP claimed
US-6008386-A ALPHA-AMINO ACIDS BEARING AN OXIRANE RING ON THE ALPHA CARBON IN PLACE OF THE ALPHA-PROTON; IRREVERSIBLE INHIBITORS FOR AMINO ACID DECARBOXYLASES BOARD OF REGENTS UNIVERSITY OF NEBRASKA-LINCOLN (US) 1999-12-28 US disclosed
US-5705660-A Method for the synthesis of α-oxiranyl amino acids BOARD OF REGENTS, UNIVERSITY OF NEBRASKA-LINCOLN 1998-01-06 US disclosed
US-5216125-A Active ester used for production of acylated amino acids SANSHIN KAGAKU KOGYO CO. LTD. (JP) 1993-06-01 US disclosed
EP-0346756-B1 PROCESS FOR PRODUCTION OF SULFONIUM COMPOUNDS MITSUBISHI GAS CHEMICAL COMPANY, INC. (JP) 1992-10-28 EP disclosed
US-5117031-A ACTIVE ESTERS USED FOR PRODUCTION OF ESTERS OR AMIDES AND PROCESS FOR PRODUCING ESTERS OR AMIDES SANSHIN KAGAKU KOGYO CO. LTD. (JP) 1992-05-26 US disclosed
EP-0245662-B1 P-HYDROXYPHENYLSULFONIUM SALTS AND THEIR USE IN THE PREPARATION OF ESTERS AND AMIDES SANSHIN KAGAKU KOGYO CO., LTD. (JP) 1991-08-07 EP disclosed
US-5021197-A Reacting a p-dialkylsulfoniophenol with a carbonyl halogenide in the presence of a secondary amine MITSUBISHI GAS CHEMICAL COMPANY, INC. (JP) 1991-06-04 US disclosed
EP-0346756-A1 Process for production of sulfonium compounds MITSUBISHI GAS CHEMICAL COMPANY, INC. (JP) 1989-12-20 EP disclosed
EP-0331988-A1 Sulfonium compounds, as well as process for producing active esters and amides used for the production of amides SANSHIN KAGAKU KOGYO CO., LTD. (JP) 1989-09-13 EP disclosed
US-4857656-A Active esters used for production of esters or amides and process for producing esters or amides SANSHIN KAGAKU KOGYO CO., LTD. (JP) 1989-08-15 US disclosed
EP-0245662-A1 p-Hydroxyphenylsulfonium salts and their use in the preparation of esters and amides SANSHIN KAGAKU KOGYO CO., LTD. (JP) 1987-11-19 EP disclosed