SCHEMBL8517573

SCHEMBL8517573

C=C[C@H]1CC[C@H](CCc2ccc(-c3ccc(F)cc3)nc2)CC1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 2/20 0.40
CYP11B2 P19099 2/20 0.40
AURKA O14965 1/20 0.40
ABL1 P00519 1/20 0.40
NTRK1 P04629 1/20 0.40
LCK P06239 1/20 0.40
CSF1R P07333 1/20 0.40
RET P07949 1/20 0.40
MET P08581 1/20 0.40
PDGFRB P09619 1/20 0.40
PIM1 P11309 1/20 0.40
PDGFRA P16234 1/20 0.40
FLT3 P36888 1/20 0.40
MAPK8 P45983 1/20 0.40
CDK8 P49336 1/20 0.40
MAP2K1 Q02750 1/20 0.40
MAP4K2 Q12851 1/20 0.40
ROCK1 Q13464 1/20 0.40
NTRK3 Q16288 1/20 0.40
MAPK14 Q16539 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8517575 1.00 CYP11B1 (0.40) CYP11B1CYP11B2AURKAABL1NTRK1
SCHEMBL8517992 0.88 MAOB (0.39) KCNH2MAOBNPC1RAB9ASMN1; SMN2
SCHEMBL8517996 0.88 MAOB (0.39) KCNH2MAOBNPC1RAB9ASMN1; SMN2
SCHEMBL8518726 0.88 CYP11B1 (0.40) CYP11B1CYP11B2AURKAABL1NTRK1
SCHEMBL9312701 0.88 CYP11B1 (0.40) CYP11B1CYP11B2AURKAABL1NTRK1
SCHEMBL8517543 0.87 NPC1 (0.44) CYP11B1CYP11B2METNPC1RAB9A
SCHEMBL8518049 0.87 NPC1 (0.44) CYP11B1CYP11B2METNPC1RAB9A
SCHEMBL9311825 0.86 AURKA (0.41) CYP11B1CYP11B2AURKAABL1NTRK1
SCHEMBL8518235 0.86 AURKA (0.41) CYP11B1CYP11B2AURKAABL1NTRK1
SCHEMBL8518233 0.86 AURKA (0.41) CYP11B1CYP11B2AURKAABL1NTRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0475273-B1 Liquid crystal mixture containing halogenated alcenyl compounds MERCK PATENT GMBH (DE) 1999-04-07 EP disclosed
US-5292452-A Electrooptical devices; high dielectric anisotropy, low rotation viscosity, short response time HOFFMANN-LA ROCHE INC. (US) 1994-03-08 US disclosed
EP-0475273-A1 Halogenated alcenyl compounds F. HOFFMANN-LA ROCHE AG (CH) 1992-03-18 EP disclosed