SCHEMBL8517868

SCHEMBL8517868

Cc1c(F)cc(-n2nnnc2C(F)(F)F)cc1Br

nearest known ligand 0.37

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.37
HTT P42858 3/20 0.37
MAPT P10636 2/20 0.37
HPGD P15428 2/20 0.37
CACNA1B Q00975 2/20 0.37
APBA1 Q02410 2/20 0.37
HSP90AA1 P07900 1/20 0.37
NOTUM Q6P988 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C19 P33261 1/20 0.35
CCR6 P51684 1/20 0.33
KCNN4 O15554 2/20 0.32
LMNA P02545 2/20 0.32
TACR1 P25103 2/20 0.31
GABRB3 P28472 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
POLB P06746 1/20 0.30
L3MBTL1 Q9Y468 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8517947 0.78 NOTUM (0.45) ALDH1A1HTTMAPTHPGDCACNA1B
SCHEMBL6541068 0.74 NOTUM (0.46) ALDH1A1HTTMAPTHPGDCACNA1B
SCHEMBL8176205 0.72 TACR1 (0.48) ALDH1A1MAPTHPGDTACR1
SCHEMBL8332932 0.72 HTT (0.36) ALDH1A1HTTMAPTHPGDCACNA1B
SCHEMBL5345569 0.71 TACR1 (0.37) ALDH1A1HTTMAPTHPGDCACNA1B
SCHEMBL8329084 0.70 ALDH1A1 (0.33) ALDH1A1HTTMAPTHPGDCACNA1B
SCHEMBL6100503 0.70 ALDH1A1 (0.47) ALDH1A1HTTMAPTHPGDCACNA1B
SCHEMBL5551503 0.70 ALDH1A1 (0.70) ALDH1A1HTTMAPTHPGDCACNA1B
SCHEMBL5935000 0.69 TACR1 (0.39) ALDH1A1HTTMAPTHPGDCACNA1B
SCHEMBL13801193 0.69 ALDH1A1 (0.43) ALDH1A1HTTMAPTHPGDCACNA1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5877191-A ANTIINFLAMMATORY AGENT; ANALGESICS; ANTIHISTAMINES; EMESIS MERCK & CO., INC. (US) 1999-03-02 US disclosed