SCHEMBL8519909

SCHEMBL8519909

CC1=NCC(=O)Nc2c(C)cccc21

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DAO P14920 1/20 0.50
HTR5A P47898 2/20 0.41
POLB P06746 1/20 0.40
PGR P06401 1/20 0.40
GABRA1 P14867 1/20 0.40
GABRG2 P18507 1/20 0.40
GABRB3 P28472 1/20 0.40
GABRA5 P31644 1/20 0.40
GABRA3 P34903 1/20 0.40
GABRA2 P47869 1/20 0.40
GABRB2 P47870 1/20 0.40
CREBBP Q92793 1/20 0.39
AGTR1 P30556 1/20 0.38
ALDH1A1 P00352 4/20 0.37
GAA P10253 2/20 0.37
MAPT P10636 2/20 0.37
PARP1 P09874 1/20 0.36
PARP10 Q53GL7 1/20 0.36
PARP11 Q9NR21 1/20 0.36
CA1 P00915 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29391065 0.76 GABRA1 (0.61) PGRGABRA1GABRG2GABRB3GABRA5
SCHEMBL3259073 0.76 GABRA1 (0.61) PGRGABRA1GABRG2GABRB3GABRA5
SCHEMBL30865023 0.75 GABRA1 (0.46) DAOGABRA1GABRG2GABRB3GABRA5
SCHEMBL28124567 0.75 GABRA1 (0.46) DAOGABRA1GABRG2GABRB3GABRA5
SCHEMBL10027162 0.74 PARP1 (0.41) PGRALDH1A1MAPTPARP1HPGD
SCHEMBL10822678 0.69 HDAC8 (0.50) DAOHTR5ACA1CA2CA7
SCHEMBL10629910 0.69 DAO (0.49) DAOPOLBCREBBPAGTR1ALDH1A1
SCHEMBL3088689 0.67 DAO (1.00) DAOPOLBAGTR1ALDH1A1GAA
Hydrochloric Acid SCHEMBL11430657 0.66 DAO (0.96) DAOPOLBAGTR1ALDH1A1GAA
SCHEMBL8561720 0.66 MEN1 (0.51) POLBGABRA1GABRG2GABRB3GABRA5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0934282-A1 1,4-BENZODIAZEPINONES AND THEIR USES AS CCK ANTAGONISTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1999-08-11 EP disclosed
WO-1998015535-A1 1,4-BENZODIAZEPINONES AND THEIR USES AS CCK ANTAGONISTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1998-04-16 WO disclosed