SCHEMBL8523959

SCHEMBL8523959

O=C(Nc1ccc2[nH]ccc2c1)c1cccnc1

nearest known ligand 0.71

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 5/20 0.71
NPC1 O15118 4/20 0.71
MAPT P10636 1/20 0.71
ALDH1A1 P00352 2/20 0.66
MEN1 O00255 1/20 0.66
KMT2A Q03164 1/20 0.66
SMN1; SMN2 Q16637 1/20 0.66
ATR Q13535 1/20 0.62
KCNK3 O14649 1/20 0.58
LMNA P02545 1/20 0.57
HIF1A Q16665 1/20 0.57
HPGD P15428 1/20 0.57
HSD17B10 Q99714 1/20 0.57
PRKCI P41743 1/20 0.56
ROCK2 O75116 1/20 0.56
ROCK1 Q13464 1/20 0.56
L3MBTL1 Q9Y468 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14082569 0.87 ATR (0.65) RAB9ANPC1MAPTALDH1A1MEN1
SCHEMBL28435041 0.84 NPC1 (0.74) RAB9ANPC1MAPTKCNK3LMNA
SCHEMBL31156451 0.84 NPC1 (1.00) RAB9ANPC1MAPTPRKCI
SCHEMBL4761937 0.84 NPC1 (1.00) RAB9ANPC1MAPTPRKCI
SCHEMBL9400611 0.83 ATR (0.57) RAB9ANPC1MAPTALDH1A1MEN1
SCHEMBL2040710 0.82 RAB9A (0.65) RAB9ANPC1ALDH1A1MEN1KMT2A
Hydrochloric Acid SCHEMBL9400692 0.82 HTR2C (0.57) RAB9ANPC1MAPTALDH1A1MEN1
SCHEMBL2569111 0.82 NPC1 (0.76) RAB9ANPC1ALDH1A1MEN1KMT2A
SCHEMBL14880457 0.80 RAB9A (1.00) RAB9ANPC1MAPTALDH1A1MEN1
SCHEMBL3931668 0.79 BRAF (0.66) NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0882040-A4 ANTAGONISTS OF GONADOTROPIN RELEASING HORMONE MERCK & CO INC (US) 1999-02-10 EP disclosed
EP-0882040-A1 ANTAGONISTS OF GONADOTROPIN RELEASING HORMONE Merck & Co., Inc. (US) 1998-12-09 EP disclosed
WO-1997021707-A1 ANTAGONISTS OF GONADOTROPIN RELEASING HORMONE MERCK & CO., INC. (US) 1997-06-19 WO disclosed