SCHEMBL8524556

SCHEMBL8524556

COC(=O)N[C@H](C(=O)N1CCC[C@H]1C(=O)NI)[C@@H](C)OC

nearest known ligand 0.44

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 2/20 0.43
CYP3A4 P08684 8/20 0.40
CYP2C9 P11712 7/20 0.40
CYP2C19 P33261 5/20 0.40
CYP2D6 P10635 2/20 0.40
CYP1A2 P05177 2/20 0.40
ELANE P08246 7/20 0.39
NR1I2 O75469 1/20 0.39
ABCB11 O95342 1/20 0.39
OPRK1 P41145 1/20 0.39
F2 P00734 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10299121 0.90 KCNH2 (0.44) KCNH2CYP3A4CYP2C9CYP2C19CYP2D6
SCHEMBL5987813 0.90 KCNH2 (0.44) KCNH2CYP3A4CYP2C9CYP2C19CYP2D6
SCHEMBL3269632 0.89 ELANE (0.44) KCNH2CYP3A4CYP2C9CYP2C19CYP2D6
SCHEMBL3268486 0.89 ELANE (0.44) KCNH2CYP3A4CYP2C9CYP2C19CYP2D6
SCHEMBL18913820 0.86 ACE (0.50) KCNH2F2
SCHEMBL21641823 0.86 ACE (0.50) KCNH2F2
SCHEMBL21641824 0.86 ACE (0.50) KCNH2F2
SCHEMBL12292177 0.86 XIAP (0.48) KCNH2CYP3A4CYP2C9CYP2C19CYP2D6
SCHEMBL18932131 0.86 FKBP5 (0.45) KCNH2CYP3A4CYP2C9CYP2C19CYP2D6
SCHEMBL18931712 0.86 FKBP5 (0.45) KCNH2CYP3A4CYP2C9CYP2C19CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2628481-A1 Trisubstituted heterocycles as replication inhibitors of hepatitis C virus HCV AbbVie Bahamas Ltd. (BS) 2013-08-21 EP disclosed
EP-2455376-A1 Heterocyclic compounds as inhibitors of hepatitis C virus (HCV) Abbott Laboratories (US) 2012-05-23 EP disclosed
WO-2010144646-A2 ANTI-VIRAL COMPOUNDS ABBOTT LABORATORIES (US) 2010-12-16 WO disclosed