SCHEMBL8524973

SCHEMBL8524973

c1ccc(CN2CCCC(c3c(-c4ccccc4)[nH]c4ccccc34)C2)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 14/20 1.00
KCNH2 Q12809 14/20 1.00
HTR2C P28335 9/20 1.00
DRD2 P14416 5/20 1.00
HDAC1 Q13547 4/20 0.69
HPGDS O60760 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8524538 0.92 HTR2A (0.84) HTR2AKCNH2HTR2CDRD2HDAC1
SCHEMBL8525084 0.88 HTR2A (1.00) HTR2AKCNH2HTR2CDRD2HDAC1
SCHEMBL10725147 0.88 KCNH2 (0.78) HTR2AKCNH2HTR2CDRD2HDAC1
SCHEMBL7955758 0.86 HTR2A (1.00) HTR2AKCNH2HTR2CDRD2HDAC1
SCHEMBL725442 0.84 KCNH2 (0.72) HTR2AKCNH2HTR2CDRD2HDAC1
SCHEMBL724547 0.83 HDAC1 (1.00) HTR2AKCNH2HTR2CDRD2HDAC1
SCHEMBL724548 0.83 HDAC1 (1.00) HTR2AKCNH2HTR2CDRD2HDAC1
SCHEMBL8525408 0.81 HTR2A (1.00) HTR2AKCNH2HTR2CDRD2HDAC1
SCHEMBL8524585 0.78 HTR2A (1.00) HTR2AKCNH2HTR2CDRD2HDAC1
SCHEMBL7647583 0.77 HTR2A (0.63) HTR2AKCNH2HTR2CDRD2HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1999047511-A1 INDOLE DERIVATIVES AS 5-HT2A RECEPTOR ANTAGONISTS MERCK SHARP & DOHME LIMITED (GB) 1999-09-23 WO claimed
WO-1999047511-A1 INDOLE DERIVATIVES AS 5-HT2A RECEPTOR ANTAGONISTS MERCK SHARP & DOHME LIMITED (GB) 1999-09-23 WO disclosed