SCHEMBL8525752

SCHEMBL8525752

CCOC(=O)c1noc(C2CC2)c1C(=O)c1ccc(-n2nccn2)cc1C(F)(F)F

nearest known ligand 0.41

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 2/20 0.41
HCRTR2 O43614 10/20 0.41
HCRTR1 O43613 6/20 0.34
HTT P42858 1/20 0.34
MLYCD O95822 1/20 0.33
CYP3A4 P08684 3/20 0.33
NPC1 O15118 1/20 0.33
ALDH1A1 P00352 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
HSP90AA1 P07900 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8486767 0.88 NR1H4 (0.41) NR1H4HCRTR2HTTNPC1ALDH1A1
SCHEMBL8525775 0.88 HCRTR2 (0.43) NR1H4HCRTR2HCRTR1HTTCYP3A4
SCHEMBL8525290 0.88 HCRTR2 (0.43) NR1H4HCRTR2HCRTR1CYP3A4ALDH1A1
SCHEMBL8525429 0.87 NR1H4 (0.40) NR1H4HTTHSP90AA1
SCHEMBL8491830 0.87 NR1H4 (0.40) NR1H4HCRTR2HTTALDH1A1
SCHEMBL8524086 0.87 NR1H4 (0.40) NR1H4HCRTR2HCRTR1HTTCYP3A4
SCHEMBL8487140 0.86 HTT (0.43) NR1H4HCRTR2HCRTR1HTTMLYCD
SCHEMBL8525770 0.85 HCRTR2 (0.41) HCRTR2HCRTR1HTTCYP3A4ALDH1A1
SCHEMBL8490491 0.85 NR1H4 (0.41) NR1H4HTTMLYCDALDH1A1
SCHEMBL8524334 0.84 HCRTR2 (0.43) HCRTR2HCRTR1MLYCDCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1999003856-A1 4-BENZOYL-ISOXAZOLE- AND -PYRAZOLE DERIVATIVES AND 2-CYANO 1,3-DIONE DERIVATIVES AS HERBICIDES RHONE-POULENC AGRICULTURE LIMITED (GB) 1999-01-28 WO disclosed