SCHEMBL8525844

SCHEMBL8525844

CCCC1(CCC)CC(=O)Nc2ccccc2C1

nearest known ligand 0.49

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
AHR P35869 1/20 0.49
PDK2 Q15119 1/20 0.49
NPC1 O15118 1/20 0.47
MAPK13 O15264 1/20 0.47
MAPK12 P53778 1/20 0.47
MAPK11 Q15759 1/20 0.47
MAPK14 Q16539 1/20 0.47
BRD4 O60885 8/20 0.45
CREBBP Q92793 6/20 0.45
MAPT P10636 1/20 0.45
CYP19A1 P11511 1/20 0.37
SRC P12931 1/20 0.37
NPSR1 Q6W5P4 1/20 0.36
ADRA2A P08913 1/20 0.36
ADRA2B P18089 1/20 0.36
ADRA2C P18825 1/20 0.36
EP300 Q09472 1/20 0.36
HTR1A P08908 2/20 0.34
GAA P10253 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8524680 0.74 AHR (0.57) AHRPDK2NPC1MAPK13MAPK12
SCHEMBL18826462 0.70 KDM4E (0.43) CYP19A1NPSR1
SCHEMBL3646873 0.69 NPSR1 (0.44) AHRPDK2NPC1BRD4CREBBP
Oxindole SCHEMBL11087237 0.69 AHR (0.78) AHRPDK2NPC1MAPK13MAPK12
Alcohol SCHEMBL10571326 0.68 NPC1 (0.79) AHRPDK2NPC1MAPK13MAPK12
SCHEMBL19289267 0.67 ADRA2A (0.41) ADRA2AHTR1A
SCHEMBL23674847 0.67 NPSR1 (0.52) AHRPDK2NPC1MAPK13MAPK12
SCHEMBL21061671 0.67 AHR (0.52) AHRPDK2NPC1MAPK13MAPK12
Oxindole SCHEMBL8866522 0.67 AHR (0.72) AHRPDK2NPC1MAPK13MAPK12
SCHEMBL30100714 0.67 NPSR1 (0.52) AHRPDK2NPC1MAPK13MAPK12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1999015524-A1 THIAZOLE DERIVATIVES FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1999-04-01 WO disclosed