SCHEMBL8525859

SCHEMBL8525859

NCCC[C@H](C(N)=O)N(Cc1ccc(CC(N)=O)cc1)C(=O)C(c1ccccc1)c1ccccc1

nearest known ligand 0.40

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.40
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
NR1H3 Q13133 3/20 0.37
EPOR P19235 2/20 0.36
HTR2A P28223 1/20 0.36
HRH1 P35367 1/20 0.36
RORC P51449 1/20 0.36
MC4R P32245 2/20 0.34
MC5R P33032 2/20 0.34
MC3R P41968 2/20 0.34
CA2 P00918 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8650060 0.92 TDP1 (0.41) TDP1MEN1KMT2AEPORHTR2A
SCHEMBL8650581 0.91 TDP1 (0.43) TDP1MEN1KMT2AEPORHTR2A
SCHEMBL8126608 0.90 TDP1 (0.41) TDP1MEN1KMT2AEPORHTR2A
SCHEMBL8119409 0.86 EPOR (0.43) TDP1MEN1KMT2AEPORMC4R
SCHEMBL8528953 0.86 TDP1 (0.41) TDP1MEN1KMT2ANR1H3RORC
SCHEMBL8127789 0.86 TDP1 (0.46) TDP1MEN1KMT2ANR1H3EPOR
SCHEMBL7039838 0.85 TDP1 (0.36) TDP1MEN1KMT2ANR1H3RORC
Hydrochloric Acid SCHEMBL8120628 0.84 EPOR (0.41) TDP1MEN1KMT2AEPORMC4R
SCHEMBL8651940 0.84 EPOR (0.56) EPOR
SCHEMBL9196210 0.82 TACR1 (0.36) TDP1MEN1KMT2AEPORHTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0885186-A1 AMINO ACID DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONTAINING THESE COMPOUNDS AND PROCESSES FOR PREPARING THEM Dr. Karl Thomae GmbH (DE) 1998-12-23 EP disclosed
WO-1997019911-A1 AMINO ACID DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONTAINING THESE COMPOUNDS AND PROCESSES FOR PREPARING THEM DR. KARL THOMAE GMBH (DE) 1997-06-05 WO disclosed