SCHEMBL8526244

SCHEMBL8526244

CCOC(=O)NC(=O)N(C)Cc1ccc(CN(C(=O)C(c2ccccc2)c2ccccc2)[C@H](CCCNC(=N)N)C(N)=O)cc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 2/20 0.38
NPY1R P25929 4/20 0.38
MEN1 O00255 3/20 0.37
KMT2A Q03164 3/20 0.37
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2C19 P33261 1/20 0.34
LMNA P02545 2/20 0.33
F2 P00734 1/20 0.33
L3MBTL1 Q9Y468 2/20 0.32
ALDH1A1 P00352 1/20 0.32
POLB P06746 1/20 0.32
HSD17B10 Q99714 1/20 0.32
HDAC3 O15379 1/20 0.32
HDAC4 P56524 1/20 0.32
HDAC1 Q13547 1/20 0.32
HDAC7 Q8WUI4 1/20 0.32
HDAC2 Q92769 1/20 0.32
HDAC10 Q969S8 1/20 0.32
HDAC11 Q96DB2 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL8529043 0.95 TDP1 (0.36) TDP1NPY1RMEN1KMT2ACYP3A4
SCHEMBL8612537 0.89 NPY1R (0.42) NPY1RMEN1KMT2ACYP3A4CYP2D6
SCHEMBL7750689 0.84 MEN1 (0.42) TDP1MEN1KMT2AF2
Trifluoroacetic Acid SCHEMBL7040972 0.84 NPY1R (0.38) NPY1RHDAC1NPFFR1
SCHEMBL7750620 0.84 KMT2A (0.41) MEN1KMT2AALDH1A1
SCHEMBL1389118 0.83 CNR1 (0.41) TDP1MEN1KMT2A
SCHEMBL30905434 0.83 CNR1 (0.41) TDP1MEN1KMT2A
SCHEMBL4651738 0.83 TDP1 (0.39) TDP1NPY1RMEN1KMT2A
SCHEMBL4653161 0.83 CNR1 (0.43) TDP1MEN1KMT2A
SCHEMBL4651831 0.82 CNR1 (0.42) TDP1NPY1RMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0885186-A1 AMINO ACID DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONTAINING THESE COMPOUNDS AND PROCESSES FOR PREPARING THEM Dr. Karl Thomae GmbH (DE) 1998-12-23 EP disclosed
WO-1997019911-A1 AMINO ACID DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONTAINING THESE COMPOUNDS AND PROCESSES FOR PREPARING THEM DR. KARL THOMAE GMBH (DE) 1997-06-05 WO disclosed