SCHEMBL8526260

SCHEMBL8526260

N=C(N)NCCC[C@H](C(N)=O)N(Cc1ccc(CNC(N)=O)cc1)C(=O)Cc1ccc(Cl)cc1Cl

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
ERCC1 P07992 5/20 0.39
ERCC4 Q92889 5/20 0.39
L3MBTL1 Q9Y468 2/20 0.36
MEN1 O00255 1/20 0.36
ALDH1A1 P00352 1/20 0.36
THRB P10828 1/20 0.36
HTT P42858 1/20 0.36
KMT2A Q03164 1/20 0.36
HDAC8 Q9BY41 3/20 0.35
TDP1 Q9NUW8 1/20 0.34
METAP2 P50579 1/20 0.34
POLB P06746 1/20 0.33
HSP90AA1 P07900 1/20 0.33
MAPT P10636 1/20 0.33
RECQL P46063 1/20 0.33
LMNA P02545 1/20 0.33
MAPK1 P28482 1/20 0.33
NLRP1 Q9C000 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL8526755 0.94 NPY4R (0.35) CYP2C9CYP2C19ERCC1ERCC4L3MBTL1
SCHEMBL8528690 0.86 CYP2C9 (0.39) CYP2C9CYP2C19MEN1HTTKMT2A
SCHEMBL8525688 0.82 NPY4R (0.38) CYP2C9CYP2C19
Trifluoroacetic Acid SCHEMBL8526744 0.81 NPY4R (0.35) CYP2C9CYP2C19HTT
Trifluoroacetic Acid SCHEMBL8527841 0.81 NPY4R (0.36) CYP2C9CYP2C19
SCHEMBL6898666 0.80 CYP2C9 (0.45) CYP2C9CYP2C19MEN1THRBKMT2A
SCHEMBL8526887 0.80 KMT2A (0.33) CYP2C9CYP2C19L3MBTL1MEN1KMT2A
SCHEMBL8585843 0.78 KMT2A (0.45) MEN1ALDH1A1KMT2AMAPTLMNA
SCHEMBL4651754 0.77 NPY4R (0.39)
SCHEMBL8125850 0.77 PTPRB (0.42) CYP2C9CYP2C19L3MBTL1ALDH1A1THRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0885186-A1 AMINO ACID DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONTAINING THESE COMPOUNDS AND PROCESSES FOR PREPARING THEM Dr. Karl Thomae GmbH (DE) 1998-12-23 EP disclosed
WO-1997019911-A1 AMINO ACID DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONTAINING THESE COMPOUNDS AND PROCESSES FOR PREPARING THEM DR. KARL THOMAE GMBH (DE) 1997-06-05 WO disclosed