SCHEMBL8528690

SCHEMBL8528690

N=C(N)NCCC[C@H](C(N)=O)N(Cc1ccc(CNC(N)=O)cc1)C(=O)Cc1c(Cl)cccc1Cl

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 2/20 0.39
CYP2C19 P33261 2/20 0.39
HTT P42858 1/20 0.33
ITGB1 P05556 1/20 0.32
ITGA5 P08648 1/20 0.32
FNTA P49354 1/20 0.32
FNTB P49356 1/20 0.32
ADRA2A P08913 2/20 0.31
MEN1 O00255 1/20 0.31
LMNA P02545 1/20 0.31
CYP3A4 P08684 1/20 0.31
HTR1A P08908 1/20 0.31
CYP2D6 P10635 1/20 0.31
ADRA2B P18089 1/20 0.31
ADRA2C P18825 1/20 0.31
MAOA P21397 1/20 0.31
ADRA1D P25100 1/20 0.31
HTR2A P28223 1/20 0.31
HTR2C P28335 1/20 0.31
MAPK1 P28482 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL8526744 0.94 NPY4R (0.35) CYP2C9CYP2C19HTTITGB1ITGA5
SCHEMBL8526260 0.86 CYP2C9 (0.40) CYP2C9CYP2C19HTTMEN1LMNA
SCHEMBL8525688 0.85 NPY4R (0.38) CYP2C9CYP2C19
Trifluoroacetic Acid SCHEMBL8526755 0.82 NPY4R (0.35) CYP2C9CYP2C19HTTMEN1LMNA
Trifluoroacetic Acid SCHEMBL8527841 0.81 NPY4R (0.36) CYP2C9CYP2C19
SCHEMBL6898666 0.80 CYP2C9 (0.45) CYP2C9CYP2C19MEN1LMNAKMT2A
SCHEMBL8526887 0.80 KMT2A (0.33) CYP2C9CYP2C19MEN1KMT2A
SCHEMBL8585843 0.78 KMT2A (0.45) FNTAFNTBMEN1LMNAKMT2A
SCHEMBL7059809 0.78 NPY1R (0.42) MEN1KMT2ATPSAB1CNR1
SCHEMBL6899868 0.78 NPY1R (0.42) MEN1KMT2ATPSAB1CNR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0885186-A1 AMINO ACID DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONTAINING THESE COMPOUNDS AND PROCESSES FOR PREPARING THEM Dr. Karl Thomae GmbH (DE) 1998-12-23 EP disclosed
WO-1997019911-A1 AMINO ACID DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONTAINING THESE COMPOUNDS AND PROCESSES FOR PREPARING THEM DR. KARL THOMAE GMBH (DE) 1997-06-05 WO disclosed