SCHEMBL8527502

SCHEMBL8527502

C1=CN=c2ccccc2=C[N]1

nearest known ligand 0.00

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Quinazoline SCHEMBL5922743 0.78
SCHEMBL5050144 0.76
SCHEMBL16690908 0.76
SCHEMBL5050151 0.76
SCHEMBL7336241 0.71
SCHEMBL25092 0.69
SCHEMBL3070232 0.65
SCHEMBL2301093 0.64
SCHEMBL5934901 0.64
SCHEMBL18935458 0.64

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0698015-A1 PREPARATION OF N-CYANODITHIOIMINO-CARBONATES AND 3-MERCAPTO-5-AMINO-1H-1,2,4-TRIAZOLE GENENTECH, INC. (US) 1996-02-28 EP claimed
WO-2013184570-A2 METHODS FOR THE SYNTHESIS OF 1,3-SUBSTITUTED AMINOURACILS AND OTHER XANTHINE-RELATED COMPOUNDS FOREST LABORATORIES HOLDINGS LIMITED (BM) 2013-12-12 WO disclosed
US-5834464-A ANXIOLYTIC AGENTS, CHOLECYSTOKININ B ANTAGONISTS MERCK & CO., INC. (US) 1998-11-10 US disclosed
US-5807875-A OBESITY THERAPY DR. KARL THOMAE GMBH (DE) 1998-09-15 US disclosed
EP-0698015-A1 PREPARATION OF N-CYANODITHIOIMINO-CARBONATES AND 3-MERCAPTO-5-AMINO-1H-1,2,4-TRIAZOLE GENENTECH, INC. (US) 1996-02-28 EP disclosed
WO-1995001970-A1 ALCOHOL TO AZIDE SN2 CONVERSION MERCK & CO., INC. (US) 1995-01-19 WO disclosed