SCHEMBL8527554

SCHEMBL8527554

CCSc1ccc2c(c1)CCN2C(C)=O

nearest known ligand 0.62

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 7/20 0.62
ALDH1A1 P00352 4/20 0.51
HPGD P15428 3/20 0.51
KDM4E B2RXH2 2/20 0.51
RECQL P46063 1/20 0.51
CYP11B1 P15538 4/20 0.48
CYP11B2 P19099 4/20 0.48
TP53 P04637 3/20 0.47
HSD17B10 Q99714 2/20 0.47
NPC1 O15118 2/20 0.47
RAB9A P51151 2/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
MAPT P10636 2/20 0.47
HTR2A P28223 1/20 0.47
HTR2C P28335 1/20 0.47
HTR2B P41595 1/20 0.47
LMNA P02545 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8528919 0.85 NOTUM (0.67) NOTUMALDH1A1HPGDKDM4ERECQL
SCHEMBL31647180 0.85 NOTUM (0.56) NOTUMALDH1A1HPGDKDM4ERECQL
SCHEMBL8526799 0.84 NOTUM (0.65) NOTUMALDH1A1HPGDKDM4ERECQL
SCHEMBL8527530 0.82 NOTUM (0.50) NOTUMALDH1A1HPGDKDM4ERECQL
SCHEMBL19777765 0.82 NOTUM (0.66) NOTUMALDH1A1HPGDKDM4ERECQL
SCHEMBL27255145 0.80 NOTUM (0.60) NOTUMALDH1A1HPGDKDM4ERECQL
SCHEMBL19777845 0.78 HTR2A (0.51) NOTUMALDH1A1KDM4ETP53HSD17B10
SCHEMBL14090157 0.78 NOTUM (0.65) NOTUMALDH1A1HPGDKDM4ERECQL
SCHEMBL5009163 0.77 NOTUM (1.00) NOTUMALDH1A1HPGDKDM4ERECQL
SCHEMBL5780390 0.75 ALDH1A1 (0.70) NOTUMALDH1A1HPGDKDM4ERECQL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5834494-A SEROTONIN 5HT2B/2C RECEPTOR ANTAGONISTS; CNS NERVOUS SYSTEM AND PSYCHOLOGICAL DISORDERS; IRRITABLE BOWEL SYNDROME SMITHKLINE BEECHAM P.L.C. (GB) 1998-11-10 US disclosed
EP-0707581-B1 INDOLINE DERIVATIVES AS 5HT2C ANTAGONISTS SMITHKLINE BEECHAM PLC (GB) 1997-02-26 EP disclosed
EP-0707581-A1 INDOLINE DERIVATIVES AS 5HT 2C? ANTAGONISTS SMITHKLINE BEECHAM PLC (GB) 1996-04-24 EP disclosed
WO-1995001976-A1 INDOLINE DERIVATIVES AS 5HT2C ANTAGONISTS SMITHKLINE BEECHAM PLC (GB) 1995-01-19 WO disclosed