SCHEMBL8528101

SCHEMBL8528101

Nc1cc(F)c(C(F)(F)F)cc1NC(=O)C(F)(F)F

nearest known ligand 0.38

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PTPN5 P54829 1/20 0.38
HDAC1 Q13547 4/20 0.36
NR3C2 P08235 1/20 0.36
CFTR P13569 4/20 0.35
AR P10275 2/20 0.35
PTGS1 P23219 2/20 0.35
L3MBTL1 Q9Y468 1/20 0.34
CA12 O43570 1/20 0.34
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
CA9 Q16790 1/20 0.34
HDAC2 Q92769 2/20 0.34
KIF11 P52732 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20051331 0.86 HDAC1 (0.40) PTPN5HDAC1PTGS1L3MBTL1CA12
SCHEMBL8530986 0.83 CFTR (0.40) PTPN5CFTRARCA12CA1
SCHEMBL4568241 0.81 PTPN5 (0.38) PTPN5ARL3MBTL1CA12CA1
SCHEMBL7750665 0.80 HDAC1 (0.36) HDAC1NR3C2ARCA1CA2
SCHEMBL6268915 0.79 CYP1A2 (0.38) PTPN5CFTRARL3MBTL1CA12
SCHEMBL22637106 0.79 HDAC1 (0.39) HDAC1NR3C2CFTRARPTGS1
SCHEMBL5396104 0.76 AR (0.44) ARL3MBTL1
SCHEMBL20051324 0.75 PTPN5 (0.38) PTPN5HDAC1L3MBTL1CA12CA1
SCHEMBL20051715 0.73 HDAC1 (0.52) HDAC1HDAC2
SCHEMBL6816450 0.72 GAA (0.47) PTPN5PTGS1L3MBTL1CA12CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0596358-B1 0-Phenylenediamines containing fluoroakyl(ene) groups and their use as intermediates in the preparation of benzimidazoles BAYER AG (DE) 1998-10-28 EP disclosed
US-5484953-A CHEMICAL INTERMEDIATES FOR BENZIMIDAZOLES FOR INSECTICIDES OR NEMATOCIDES BAYER AKTIENGESELLSCHAFT (DE) 1996-01-16 US disclosed
EP-0596358-A1 0-Phenylenediamines containing fluoroakyl(ene) groups and their use as intermediates in the preparation of benzimidazoles BAYER AG (DE) 1994-05-11 EP disclosed