SCHEMBL8530986

SCHEMBL8530986

Nc1cc(Br)c(C(F)(F)F)cc1NC(=O)C(F)(F)F

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CFTR P13569 7/20 0.40
NOTUM Q6P988 1/20 0.38
MAPT P10636 3/20 0.38
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
NPSR1 Q6W5P4 2/20 0.38
LMNA P02545 2/20 0.38
PTPN5 P54829 1/20 0.38
XBP1 P17861 1/20 0.38
AR P10275 1/20 0.37
CA2 P00918 2/20 0.36
CA12 O43570 1/20 0.36
CA1 P00915 1/20 0.36
CA9 Q16790 1/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
HTT P42858 2/20 0.36
EPHX1 P07099 1/20 0.36
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
TAS2R14 Q9NYV8 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8528101 0.83 PTPN5 (0.38) CFTRPTPN5ARCA2CA12
SCHEMBL8134148 0.81 F2R (0.40) CFTRNOTUMMAPTMEN1KMT2A
SCHEMBL15103066 0.79 MAPT (0.40) NOTUMMAPTMEN1KMT2ANPSR1
SCHEMBL6268915 0.78 CYP1A2 (0.38) CFTRMEN1KMT2ALMNAPTPN5
SCHEMBL1797636 0.77 AR (0.43) MAPTMEN1KMT2ALMNAAR
SCHEMBL4568241 0.76 PTPN5 (0.38) NOTUMMAPTMEN1KMT2ANPSR1
SCHEMBL4568240 0.75 SMN1; SMN2 (0.41) NOTUMMAPTMEN1KMT2ANPSR1
SCHEMBL4568242 0.75 KDR (0.43) MEN1KMT2ALMNAPTPN5CA2
SCHEMBL12763858 0.75 CFTR (0.39) CFTRNOTUMMAPTMEN1KMT2A
SCHEMBL29896845 0.75 CFTR (0.39) CFTRNOTUMMAPTMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0596358-B1 0-Phenylenediamines containing fluoroakyl(ene) groups and their use as intermediates in the preparation of benzimidazoles BAYER AG (DE) 1998-10-28 EP disclosed
US-5484953-A CHEMICAL INTERMEDIATES FOR BENZIMIDAZOLES FOR INSECTICIDES OR NEMATOCIDES BAYER AKTIENGESELLSCHAFT (DE) 1996-01-16 US disclosed
EP-0596358-A1 0-Phenylenediamines containing fluoroakyl(ene) groups and their use as intermediates in the preparation of benzimidazoles BAYER AG (DE) 1994-05-11 EP disclosed