SCHEMBL8528686

SCHEMBL8528686

CC(=O)Nc1ccc(C(O)C(C)CCl)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.50
TP53 P04637 1/20 0.50
HIF1A Q16665 1/20 0.50
AKR1C3 P42330 1/20 0.48
AKR1C1 Q04828 1/20 0.48
KMT2A Q03164 6/20 0.47
MEN1 O00255 5/20 0.47
SMN1; SMN2 Q16637 3/20 0.47
CYP2C19 P33261 2/20 0.47
HPGD P15428 2/20 0.47
RAB9A P51151 2/20 0.47
KDM4E B2RXH2 1/20 0.47
HTT P42858 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
DHODH Q02127 1/20 0.47
TSHR P16473 2/20 0.46
TDP1 Q9NUW8 2/20 0.46
MAPT P10636 2/20 0.46
CA12 O43570 1/20 0.46
BRD4 O60885 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4047496 0.81 SMN1; SMN2 (0.55) ALDH1A1AKR1C3AKR1C1KMT2AMEN1
SCHEMBL14463078 0.77 SMN1; SMN2 (0.59) ALDH1A1AKR1C3AKR1C1KMT2AMEN1
SCHEMBL4986450 0.77 SMN1; SMN2 (0.50) ALDH1A1TP53HIF1AAKR1C3AKR1C1
SCHEMBL4048000 0.75 ALDH1A1 (0.53) ALDH1A1AKR1C3AKR1C1KMT2AMEN1
SCHEMBL104524 0.75 SMN1; SMN2 (0.61) ALDH1A1AKR1C3AKR1C1KMT2AMEN1
SCHEMBL11112670 0.75 SMN1; SMN2 (0.61) ALDH1A1AKR1C3AKR1C1KMT2AMEN1
SCHEMBL27254651 0.73 SMN1; SMN2 (0.64) ALDH1A1AKR1C3AKR1C1KMT2AMEN1
SCHEMBL9893031 0.73 TSHR (0.73) ALDH1A1TP53KMT2AMEN1SMN1; SMN2
SCHEMBL2700912 0.73 SMN1; SMN2 (0.53) ALDH1A1AKR1C3AKR1C1KMT2AMEN1
SCHEMBL28638974 0.72 ALDH1A1 (0.60) ALDH1A1TP53HIF1AKMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5830875-A PARASITICIDES MERCK & CO., INC. (US) 1998-11-03 US disclosed
US-5208222-A Anthelemetic MERCK & CO., INC. (US) 1993-05-04 US disclosed
EP-0506331-A1 4\"-and 4'-alkylthio-avermectin derivatives MERCK & CO. INC. (US) 1992-09-30 EP disclosed
EP-0428286-A2 24- and 25-substituted avermectin and milbemycin derivatives MERCK & CO. INC. (US) 1991-05-22 EP disclosed