SCHEMBL8529993

SCHEMBL8529993

CCCCC(=O)O[C@H]1[C@H](O)[C@@H](CO)O[C@H]1n1cnc2c(OC)nc(N)nc21

nearest known ligand 0.53

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
SLC29A1 Q99808 4/20 0.53
ADORA2A P29274 4/20 0.50
ADORA2B P29275 4/20 0.50
CYP2C19 P33261 1/20 0.49
ADORA3 P0DMS8 1/20 0.49
ADORA1 P30542 1/20 0.49
TK2 O00142 2/20 0.47
PGK1 P00558 1/20 0.47
PGK2 P07205 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8530540 0.88 CYP2C19 (0.54) SLC29A1ADORA2AADORA2BCYP2C19ADORA3
SCHEMBL9019466 0.87 SLC29A1 (0.50) SLC29A1ADORA2AADORA2BADORA3ADORA1
SCHEMBL8530012 0.86 ADORA2A (0.59) SLC29A1ADORA2AADORA2BCYP2C19ADORA3
SCHEMBL8532515 0.85 CYP2C19 (0.52) SLC29A1ADORA2AADORA2BCYP2C19ADORA3
SCHEMBL17485744 0.83 HINT1 (0.56) ADORA2AADORA2BTK2
SCHEMBL8529895 0.83 P2RY11 (0.54) SLC29A1ADORA2AADORA2BCYP2C19ADORA3
SCHEMBL8529229 0.83 HINT1 (0.59) SLC29A1ADORA2AADORA2BCYP2C19ADORA3
Nelarabine SCHEMBL13575801 0.81 CYP2C19 (0.71) SLC29A1ADORA2AADORA2BCYP2C19ADORA3
Nelarabine SCHEMBL18321891 0.81 CYP2C19 (0.71) SLC29A1ADORA2AADORA2BCYP2C19ADORA3
Nelarabine SCHEMBL18820 0.81 CYP2C19 (0.71) SLC29A1ADORA2AADORA2BCYP2C19ADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5821236-A Tumor treatment with arabinofuranosyl purine derivatives GLAXO WELLCOME INC. (US) 1998-10-13 US disclosed
US-5747472-A ANTICARCINOGENIC AGENTS AND ANTITUMOR AGENTS GLAXO WELLCOME INC. (US) 1998-05-05 US disclosed
US-5492897-A ANTITUMOR AGENTS, AUTOIMMUNE DISEASES BURROUGHS WELLCOME CO. (141) (US) 1996-02-20 US disclosed
US-5424295-A Useful in treatment of varicella-zoster virus infections BURROUGHS WELLCOME CO. (US) 1995-06-13 US disclosed