SCHEMBL8530675

SCHEMBL8530675

Cc1[nH]c2ccccc2c1CC(NC(=O)OC(C)(C)C)C(=O)O

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACE P12821 2/20 0.52
PTPN1 P18031 1/20 0.51
CTSS P25774 4/20 0.49
CTSK P43235 3/20 0.49
CTSL P07711 2/20 0.49
MAPT P10636 3/20 0.49
KDM4E B2RXH2 1/20 0.49
ALDH1A1 P00352 1/20 0.49
GAA P10253 1/20 0.49
CASP1 P29466 1/20 0.49
CASP7 P55210 1/20 0.49
SCN9A Q15858 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
TACR1 P25103 2/20 0.47
TP53 P04637 1/20 0.47
PPARA Q07869 5/20 0.47
PPARG P37231 4/20 0.47
IDO1 P14902 1/20 0.46
SSTR3 P32745 1/20 0.46
PPARD Q03181 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28676764 1.00 ACE (0.52) ACEPTPN1CTSSCTSKCTSL
SCHEMBL14164211 0.90 TACR1 (0.52) ACEPTPN1CTSSCTSKCTSL
SCHEMBL6160719 0.90 ACE (0.46) ACEPTPN1CTSSCTSKCTSL
SCHEMBL6160724 0.90 ACE (0.46) ACEPTPN1CTSSCTSKCTSL
SCHEMBL6853465 0.89 TACR1 (0.52) ACECTSSCTSKCTSLMAPT
SCHEMBL26996502 0.86 MAPT (0.48) ACECTSSCTSKCTSLMAPT
SCHEMBL23127318 0.84 ATM (0.56) ACEPTPN1CTSSCTSKCTSL
SCHEMBL28556906 0.84 ATM (0.56) ACEPTPN1CTSSCTSKCTSL
SCHEMBL6854583 0.84 MAPT (0.46) CTSSCTSKCTSLMAPTKDM4E
SCHEMBL27514965 0.84 ACE (0.42) ACEPTPN1CTSSCTSKCTSL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5804578-A USEFUL FOR TREATING OSTEOPROSIS, CATABOLIC ILLNESS, IMMUNE DEFICIENCY, BONE FRACTURE, SHROT STATURE IN CHILDREN, OBASITY, SLEEP DISORDER, CACHEXIA AND PROTEIN LOSS DUE TO CHRONIC ILLNESS SUCH AS AIDS AND CANCER MERCK & CO., INC. (US) 1998-09-08 US disclosed