SCHEMBL6160724

SCHEMBL6160724

Cc1[nH]c2ccccc2c1CC(NC(=O)C(C)(C)NC(=O)OC(C)(C)C)C(=O)O

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACE P12821 3/20 0.46
MAPT P10636 3/20 0.44
KDM4E B2RXH2 1/20 0.44
ALDH1A1 P00352 1/20 0.44
GAA P10253 1/20 0.44
CASP1 P29466 1/20 0.44
CASP7 P55210 1/20 0.44
CTSL P07711 1/20 0.43
CTSS P25774 1/20 0.43
CTSK P43235 1/20 0.43
SCN9A Q15858 1/20 0.42
PTPN1 P18031 1/20 0.42
SSTR3 P32745 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
TACR1 P25103 2/20 0.41
TP53 P04637 1/20 0.41
ALOX15 P16050 1/20 0.41
EGFR P00533 1/20 0.39
SRC P12931 1/20 0.39
MEN1 O00255 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6160719 1.00 ACE (0.46) ACEMAPTKDM4EALDH1A1GAA
SCHEMBL28676764 0.90 ACE (0.52) ACEMAPTKDM4EALDH1A1GAA
SCHEMBL8530675 0.90 ACE (0.52) ACEMAPTKDM4EALDH1A1GAA
SCHEMBL6163772 0.83 KMT2A (0.43) SMN1; SMN2MEN1KMT2A
SCHEMBL6163768 0.83 KMT2A (0.43) SMN1; SMN2MEN1KMT2A
SCHEMBL27514965 0.82 ACE (0.42) ACEMAPTKDM4EALDH1A1GAA
SCHEMBL6160817 0.82 MAPT (0.50) ACEMAPTKDM4EALDH1A1GAA
SCHEMBL6160808 0.82 MAPT (0.50) ACEMAPTKDM4EALDH1A1GAA
SCHEMBL5253098 0.82 ACE (0.70) ACEMAPTCTSLCTSSCTSK
SCHEMBL5253093 0.82 ACE (0.70) ACEMAPTCTSLCTSSCTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0828754-B1 DIPEPTIDES WHICH PROMOTE RELEASE OF GROWTH HORMONE PFIZER (US) 2005-02-02 EP disclosed
US-5936089-A PIPERIDINE DERIVATIVES; BONE DISORDERS; OBESITY; AGING; CACHEXIA ASSOCIATED WITH AIDS AND CANCER PFIZER INC (US) 1999-08-10 US disclosed
EP-0828754-A1 DIPEPTIDES WHICH PROMOTE RELEASE OF GROWTH HORMONE PFIZER INC. (US) 1998-03-18 EP disclosed
CN-1143647-A Dipeptides which promote release of growth hormone PFIZER (US) 1997-02-26 CN disclosed
WO-1996038471-A1 DIPEPTIDES WHICH PROMOTE RELEASE OF GROWTH HORMONE PFIZER INC. (US) 1996-12-05 WO disclosed