SCHEMBL8531237

SCHEMBL8531237

COc1ccc(OC)c2c1COC(C#N)C2

nearest known ligand 0.46

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ADRA1A P35348 4/20 0.46
ACHE P22303 3/20 0.36
IMPDH2 P12268 1/20 0.34
IMPDH1 P20839 1/20 0.34
KDM4E B2RXH2 1/20 0.34
USP2 O75604 1/20 0.34
ALDH1A1 P00352 1/20 0.34
AR P10275 2/20 0.33
CYP1A2 P05177 1/20 0.33
DRD2 P14416 2/20 0.32
DRD1 P21728 2/20 0.32
PTPRF P10586 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8531892 0.72 ADRA1A (0.41) ADRA1AACHEIMPDH2IMPDH1KDM4E
SCHEMBL8530552 0.71 ADRA1A (0.47) ADRA1AACHEKDM4EALDH1A1DRD2
SCHEMBL8527998 0.71 ADRA1A (0.47) ADRA1AACHEKDM4EALDH1A1CYP1A2
SCHEMBL8529815 0.70 ADRA1A (0.46) ADRA1AACHEKDM4EALDH1A1CYP1A2
SCHEMBL8528876 0.70 ADRA1A (0.46) ADRA1AACHEKDM4EALDH1A1CYP1A2
SCHEMBL8528043 0.70 ADRA1A (0.46) ADRA1AACHEKDM4EALDH1A1CYP1A2
SCHEMBL8903286 0.70 ADRA1A (0.46) ADRA1AACHEKDM4EALDH1A1CYP1A2
SCHEMBL27354246 0.70 ADRA1A (0.46) ADRA1AACHEKDM4EALDH1A1CYP1A2
SCHEMBL8528366 0.69 ADRA1A (0.44) ADRA1AACHEKDM4EUSP2ALDH1A1
SCHEMBL8527470 0.69 CYP1A2 (0.47) ADRA1AACHEALDH1A1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5606037-A Processes antineoplastic heteronaphthoquinones BIOCHEM PHARMA INC. (CA) 1997-02-25 US claimed
US-5736523-A ADMINISTERING TO THE MAMMAL SUFFERING FROM CANCER BIOCHEM PHARMA INC. (CA) 1998-04-07 US disclosed
US-5606037-A Processes antineoplastic heteronaphthoquinones BIOCHEM PHARMA INC. (CA) 1997-02-25 US disclosed
EP-0659190-A1 ANTINEOPLASTIC HETERONAPHTHOQUINONES BIOCHEM PHARMA INC (CA) 1995-06-28 EP disclosed
WO-1994011382-A1 ANTINEOPLASTIC HETERONAPHTHOQUINONES BIOCHEM PHARMA INC. (CA) 1994-05-26 WO disclosed