SCHEMBL8534390

SCHEMBL8534390

CCC(=O)c1cnn(Cc2ccc(OC(F)(F)F)cc2)c1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KLKB1 P03952 3/20 0.55
TSHR P16473 1/20 0.44
CACNA1H O95180 3/20 0.43
CACNA1G O43497 2/20 0.43
CACNA1I Q9P0X4 2/20 0.43
GRIN1 Q05586 1/20 0.42
GRIN2B Q13224 1/20 0.42
PPARD Q03181 1/20 0.42
PPARA Q07869 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
AADAT Q8N5Z0 1/20 0.41
GCGR P47871 1/20 0.41
ALDH1A1 P00352 1/20 0.41
HSD17B10 Q99714 1/20 0.41
ABL1 P00519 1/20 0.41
BCR P11274 1/20 0.41
LSS P48449 1/20 0.41
PDE2A O00408 1/20 0.41
SERPINE1 P05121 1/20 0.40
BCHE P06276 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8532976 0.91 KLKB1 (0.53) KLKB1TSHRCACNA1HCACNA1GCACNA1I
SCHEMBL18987207 0.88 KLKB1 (0.44) KLKB1L3MBTL1GCGRABL1PDE2A
SCHEMBL18987058 0.87 KLKB1 (0.52) KLKB1CACNA1HCACNA1GCACNA1IGRIN1
SCHEMBL2819900 0.87 KLKB1 (0.56) KLKB1TSHRCACNA1HCACNA1GCACNA1I
SCHEMBL2511099 0.85 L3MBTL1 (0.56) KLKB1GRIN1GRIN2BL3MBTL1HSD17B10
SCHEMBL27844387 0.82 MAPT (0.56) KLKB1GRIN1GRIN2BALDH1A1HSD17B10
SCHEMBL21910761 0.81 MAPT (0.45) KLKB1GRIN1GRIN2BL3MBTL1ALDH1A1
SCHEMBL20250854 0.79 CREBBP (0.54) KLKB1GRIN1GRIN2BL3MBTL1ALDH1A1
SCHEMBL2509415 0.78 L3MBTL1 (0.52) KLKB1GRIN1GRIN2BL3MBTL1
SCHEMBL19002057 0.78 KLKB1 (0.48) KLKB1TSHRAADATALDH1A1PDE2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012069856-A1 ANTIMALARIAL COMPOUNDS LIVERPOOL SCHOOL OF TROPICAL MEDICINE (GB) 2012-05-31 WO disclosed
WO-2012069856-A1 ANTIMALARIAL COMPOUNDS LIVERPOOL SCHOOL OF TROPICAL MEDICINE (GB) 2012-05-31 WO disclosed