SCHEMBL8535575

SCHEMBL8535575

CCOC(=O)C1CCC(=O)N1Cc1ccccc1

nearest known ligand 0.55

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.55
ALDH1A1 P00352 2/20 0.50
P2RX7 Q99572 2/20 0.50
GAA P10253 1/20 0.50
USP2 O75604 1/20 0.49
CYP3A4 P08684 1/20 0.48
CYP2C9 P11712 1/20 0.48
CYP2C19 P33261 1/20 0.48
ADRA1A P35348 1/20 0.48
MEN1 O00255 2/20 0.47
CAPN1 P07384 1/20 0.47
HDAC1 Q13547 1/20 0.47
HDAC6 Q9UBN7 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5166634 1.00 KMT2A (0.55) KMT2AALDH1A1P2RX7GAAUSP2
SCHEMBL28663248 0.88 FKBP1A (0.53) KMT2AP2RX7CAPN1HDAC1HDAC6
SCHEMBL21869824 0.88 FKBP1A (0.53) KMT2AP2RX7CAPN1HDAC1HDAC6
SCHEMBL6997222 0.87 GAA (0.58) KMT2AALDH1A1P2RX7GAACYP2C9
SCHEMBL21869747 0.86 KMT2A (0.62) KMT2AALDH1A1GAACYP3A4CYP2C9
SCHEMBL21869798 0.86 KMT2A (0.62) KMT2AALDH1A1GAACYP3A4CYP2C9
SCHEMBL28663232 0.86 KMT2A (0.62) KMT2AALDH1A1GAACYP3A4CYP2C9
SCHEMBL24434796 0.86 KMT2A (0.57) KMT2AALDH1A1P2RX7GAACYP3A4
SCHEMBL927807 0.86 KMT2A (0.57) KMT2AALDH1A1P2RX7GAACYP3A4
SCHEMBL2583749 0.86 KMT2A (0.57) KMT2AALDH1A1P2RX7GAACYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5817651-A ANALGESICS, RHEUMATIC DISEASES, ANTIINFLAMMATORY AGENTS SANOFI (FR) 1998-10-06 US disclosed
US-5607933-A METHODS FOR TREATMENT OF GLAUCOMA AND FOR RELIEF OF PAIN AND RHEUMATIC AND INFLAMMATORY CONDITIONS BY ADMINISTERING THE INDOLES; N-HETERYL IS 2-PIPERAZINYL STERLING WINTHROP INC. (US) 1997-03-04 US disclosed
US-5068234-A Analgesics, rheumatic diseases, antiinflammatory agents or antiglaucoma STERLING DRUG INC. (US) 1991-11-26 US disclosed
EP-0444451-A2 3-Arylcarbonyl-1H-indoles useful as therapeutic agents STERLING WINTHROP INC. (US) 1991-09-04 EP disclosed