SCHEMBL8535634

SCHEMBL8535634

O=C(NCc1ccccc1)[C@@H]1CCCN1C(=O)C1CCCN1

nearest known ligand 0.59

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.59
CYP3A4 P08684 1/20 0.59
CYP2C9 P11712 1/20 0.59
PKM P14618 1/20 0.59
CYP2C19 P33261 1/20 0.59
POLB P06746 2/20 0.56
FKBP1A P62942 3/20 0.55
HTR2C P28335 1/20 0.55
HTR2B P41595 1/20 0.55
GAA P10253 1/20 0.54
NPC1 O15118 1/20 0.53
F2 P00734 2/20 0.53
MEN1 O00255 1/20 0.50
KMT2A Q03164 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8393443 1.00 ALDH1A1 (0.59) ALDH1A1CYP3A4CYP2C9PKMCYP2C19
SCHEMBL30179363 1.00 ALDH1A1 (0.59) ALDH1A1CYP3A4CYP2C9PKMCYP2C19
Hydrochloric Acid SCHEMBL27541627 0.99 ALDH1A1 (0.58) ALDH1A1CYP3A4CYP2C9PKMCYP2C19
Glycine SCHEMBL28382745 0.95 ALDH1A1 (0.54) ALDH1A1CYP3A4CYP2C9PKMCYP2C19
Trifluoroacetic Acid SCHEMBL4372721 0.94 ALDH1A1 (0.56) ALDH1A1CYP3A4CYP2C9PKMCYP2C19
Trifluoroacetic Acid SCHEMBL4376564 0.94 ALDH1A1 (0.56) ALDH1A1CYP3A4CYP2C9PKMCYP2C19
Hydrochloric Acid SCHEMBL9275345 0.88 POLB (0.57) ALDH1A1CYP3A4CYP2C9PKMCYP2C19
Hydrochloric Acid SCHEMBL9275339 0.88 POLB (0.57) ALDH1A1CYP3A4CYP2C9PKMCYP2C19
SCHEMBL12658484 0.87 HTR2C (0.48) ALDH1A1CYP3A4CYP2C9PKMCYP2C19
SCHEMBL13263366 0.87 HTR2C (0.48) ALDH1A1CYP3A4CYP2C9PKMCYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0832104-A1 NOVEL DOLASTATIN DERIVATIVES, THEIR PREPARATION AND USE BASF AKTIENGESELLSCHAFT (DE) 1998-04-01 EP disclosed
WO-1996040751-A1 NOVEL DOLASTATIN DERIVATIVES, THEIR PREPARATION AND USE BASF AKTIENGESELLSCHAFT (DE) 1996-12-19 WO disclosed