SCHEMBL8535895

SCHEMBL8535895

Oc1ccc(-c2ncc[nH]2)cc1Cl

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NISCH Q9Y2I1 2/20 0.49
KDM4E B2RXH2 2/20 0.47
ALDH1A1 P00352 2/20 0.47
MTOR P42345 1/20 0.47
ADK P55263 1/20 0.47
ESR2 Q92731 3/20 0.46
RIPK1 Q13546 1/20 0.46
SMPD3 Q9NY59 1/20 0.45
ESR1 P03372 2/20 0.42
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP19A1 P11511 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
PDE3B Q13370 1/20 0.40
PDE3A Q14432 1/20 0.40
TSHR P16473 1/20 0.39
HSD17B10 Q99714 1/20 0.39
HSD17B1 P14061 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1923405 0.84 NISCH (0.53) NISCHKDM4EALDH1A1MTORADK
SCHEMBL1719454 0.84 NISCH (0.53) NISCHKDM4EALDH1A1MTORADK
SCHEMBL8541165 0.80 NISCH (0.53) NISCHKDM4EALDH1A1MTORADK
SCHEMBL28829248 0.79 NISCH (0.49) NISCHKDM4EALDH1A1MTORADK
SCHEMBL1688469 0.79 NISCH (0.49) NISCHKDM4EALDH1A1MTORADK
SCHEMBL8536727 0.79 ALDH1A1 (0.52) NISCHKDM4EALDH1A1MTORADK
SCHEMBL28067582 0.79 NISCH (0.49) NISCHKDM4EALDH1A1MTORADK
SCHEMBL20667462 0.78 ADORA2A (0.64) KDM4EALDH1A1ESR2RIPK1ESR1
SCHEMBL5803059 0.76 SMPD3 (0.69) NISCHKDM4EALDH1A1RIPK1SMPD3
SCHEMBL6002654 0.76 SMPD3 (0.56) NISCHKDM4EALDH1A1MTORADK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0857171-A2 IMIDAZOLE DERIVATIVES AND THE USE THEREOF AS NITROGEN MONOXIDE SYNTHASE INHIBITORS SCHERING AKTIENGESELLSCHAFT (DE) 1998-08-12 EP disclosed
WO-1997015555-A2 IMIDAZOLE DERIVATIVES AND THE USE THEREOF AS NITROGEN MONOXIDE SYNTHASE INHIBITORS SCHERING AKTIENGESELLSCHAFT (DE) 1997-05-01 WO disclosed