SCHEMBL8536371

SCHEMBL8536371

CC(C)[C@H](NC(=O)C(Cc1ccccc1)Cn1ccnc1)C(=O)O

nearest known ligand 0.58

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 1/20 0.58
MME P08473 3/20 0.50
AGTR2 P50052 3/20 0.47
ECE1 P42892 2/20 0.47
PADI4 Q9UM07 1/20 0.46
ALDH1A1 P00352 1/20 0.45
HPGD P15428 1/20 0.45
DUSP3 P51452 1/20 0.45
PTPN5 P54829 1/20 0.45
PTPN11 Q06124 1/20 0.45
LTA4H P09960 2/20 0.44
CYP19A1 P11511 1/20 0.44
CYP26A1 O43174 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9556665 0.89 HRH4 (0.60) HRH4MMEAGTR2ECE1PADI4
SCHEMBL7381214 0.84 HRH4 (0.58) HRH4MMEAGTR2ECE1PADI4
SCHEMBL7305090 0.82 HRH4 (0.61) HRH4AGTR2CYP19A1
SCHEMBL9556789 0.82 HRH4 (0.61) HRH4AGTR2CYP19A1
SCHEMBL7305085 0.82 HRH4 (0.61) HRH4AGTR2CYP19A1
SCHEMBL7382301 0.81 HRH4 (0.54) HRH4MMEPADI4
SCHEMBL9556344 0.77 HRH4 (0.58) HRH4CYP19A1
SCHEMBL8532853 0.75 HRH4 (0.60) HRH4CYP19A1CYP26A1
SCHEMBL6451863 0.72 MME (0.54) MMEECE1ALDH1A1LTA4H
SCHEMBL6451867 0.72 MME (0.54) MMEECE1ALDH1A1LTA4H

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5712417-A Inhibitors of retroviral proteases ABBOTT LABORATORIES (US) 1998-01-27 US disclosed
EP-0428849-A2 Retroviral protease inhibitors HOECHST AKTIENGESELLSCHAFT (DE) 1991-05-29 EP disclosed