SCHEMBL8536588

SCHEMBL8536588

COc1ccc(N(C)Br)cc1OC

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA2 P00918 2/20 0.52
CA12 O43570 1/20 0.52
CA1 P00915 1/20 0.52
CA7 P43166 1/20 0.52
CA9 Q16790 1/20 0.52
CA14 Q9ULX7 1/20 0.52
NQO2 P16083 2/20 0.50
ACHE P22303 1/20 0.46
ALDH1A1 P00352 3/20 0.44
CYP2C9 P11712 2/20 0.44
CYP2C19 P33261 2/20 0.44
CYP1A2 P05177 2/20 0.44
CYP3A4 P08684 2/20 0.44
HPGD P15428 1/20 0.44
BACE1 P56817 1/20 0.44
HSD17B10 Q99714 1/20 0.44
CYP2D6 P10635 1/20 0.44
BLM P54132 1/20 0.43
PMP22 Q01453 1/20 0.43
MAOA P21397 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1107760 0.82 NQO2 (0.63) CA2CA12CA1CA7CA9
SCHEMBL8943682 0.79 CA2 (0.58) CA2CA12CA1CA7CA9
SCHEMBL6887297 0.78 CA2 (0.52) CA2CA12CA1CA7CA9
SCHEMBL12320129 0.78 CA2 (0.52) CA2CA12CA1CA7CA9
SCHEMBL11662793 0.75 CA2 (0.48) CA2CA12CA1CA7CA9
SCHEMBL973685 0.75 CA2 (0.48) CA2CA12CA1CA7CA9
SCHEMBL17854040 0.75 CA2 (0.48) CA2CA12CA1CA7CA9
Hydrochloric Acid SCHEMBL3657273 0.74 BLM (0.47) CA2CA12CA1CA7CA9
SCHEMBL4859689 0.74 CSF1R (0.49) CA2CA12CA1CA7CA9
SCHEMBL8943818 0.72 CA2 (0.61) CA2CA12CA1CA7CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5721233-A Derivatives of 2,3-dihydro benzofuranols MERRELL PHARMACEUTICALS INC. (US) 1998-02-24 US disclosed
EP-0635009-B1 NOVEL DERIVATIVES OF 2,3-DIHYDRO-2,2,4,6,7-PENTAALKYL-5-BENZOFURANOLS MERRELL PHARMA INC (US) 1997-09-17 EP disclosed
EP-0635009-A1 NOVEL DERIVATIVES OF 2,3-DIHYDRO-2,2,4,6,7-PENTAALKYL-5-BENZOFURANOLS. MERRELL DOW PHARMA (US) 1995-01-25 EP disclosed
WO-1993020057-A1 NOVEL DERIVATIVES OF 2,3-DIHYDRO-2,2,4,6,7-PENTAALKYL-5-BENZOFURANOLS MERRELL DOW PHARMACEUTICALS INC. (US) 1993-10-14 WO disclosed