SCHEMBL8536815

SCHEMBL8536815

O=C(O)Cn1c(-c2ccccc2Cl)ccc(NC(=O)OCc2ccccc2)c1=O

nearest known ligand 0.67

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ELANE P08246 16/20 0.67
CTRC Q99895 3/20 0.51
CASP1 P29466 1/20 0.45
PTPN1 P18031 1/20 0.45
CASP3 P42574 1/20 0.45
NPC1 O15118 1/20 0.44
RAB9A P51151 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7445689 0.88 ELANE (0.60) ELANECTRCCASP1PTPN1CASP3
SCHEMBL1329615 0.87 ELANE (0.65) ELANECTRC
SCHEMBL8531683 0.87 ELANE (0.59) ELANECTRCCASP1PTPN1CASP3
SCHEMBL2279465 0.86 ELANE (0.58) ELANECTRCCASP1PTPN1CASP3
SCHEMBL7276488 0.85 ELANE (0.64) ELANECTRCCASP1PTPN1NPC1
SCHEMBL7402310 0.85 ELANE (0.60) ELANECTRCCASP1PTPN1CASP3
SCHEMBL21685578 0.84 NPC1 (0.50) ELANECTRCCASP1PTPN1CASP3
SCHEMBL7276654 0.81 ELANE (1.00) ELANECTRC
SCHEMBL8536676 0.81 ELANE (0.59) ELANECTRC
SCHEMBL7276644 0.80 ELANE (0.76) ELANECTRC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5721222-A Heterocyclic ketones ZENECA LIMITED (GB) 1998-02-24 US disclosed
US-5486529-A Certain pyridyl ketones for treating diseases involving leukocyte elastase ZENECA LIMITED (GB) 1996-01-23 US disclosed